SCHEMBL11245253

SCHEMBL11245253

OC(C#CI)(c1ccccc1Cl)c1ccc(Cl)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
TSHR P16473 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
MAPK1 P28482 1/20 0.46
CASR P41180 1/20 0.37
CYP19A1 P11511 2/20 0.36
CYP3A5 P20815 1/20 0.35
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.32
KCNN4 O15554 1/20 0.32
TP53 P04637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
ADRA1A P35348 1/20 0.31
OPRK1 P41145 1/20 0.31
KCNH2 Q12809 1/20 0.31
GABRA1 P14867 2/20 0.30
GABRG2 P18507 2/20 0.30
GABRB3 P28472 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11239589 0.84 CYP3A4 (0.46) CYP3A4TSHRTDP1MAPK1CASR
SCHEMBL11261677 0.83 TSHR (0.43) CYP3A4TSHRTDP1MAPK1CASR
SCHEMBL11248026 0.83 CYP19A1 (0.47) CYP3A4TSHRMAPK1CYP19A1CYP3A5
SCHEMBL11249211 0.82 CYP19A1 (0.40) CYP3A4TSHRTDP1MAPK1CASR
SCHEMBL11258277 0.78 CYP19A1 (0.42) CYP3A4TSHRTDP1MAPK1CASR
SCHEMBL11571703 0.76 TSHR (0.47) CYP3A4TSHRTDP1MAPK1CASR
SCHEMBL11247324 0.74 CYP19A1 (0.35) CYP3A4CYP19A1CYP3A5KCNN4HTR2A
SCHEMBL11869739 0.72 TSHR (0.65) CYP3A4TSHRTDP1MAPK1CASR
SCHEMBL17383651 0.68 TSHR (0.48) CYP3A4TSHRTDP1MAPK1CASR
SCHEMBL11250352 0.68 CYP19A1 (0.36) CYP3A4TSHRCYP19A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4322442-A INSECTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1982-03-30 US disclosed