SCHEMBL11246121

SCHEMBL11246121

O=C(NCc1cccc2c(C3CCCC3)nccc12)C(Cl)Cl

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NMT1 P30419 1/20 0.40
DGAT2 Q96PD7 1/20 0.37
P2RX7 Q99572 6/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
CDK5 Q00535 1/20 0.35
KLKB1 P03952 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CHRNA7 P36544 1/20 0.33
PTGES O14684 1/20 0.33
CYP3A4 P08684 1/20 0.33
ANPEP P15144 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11269174 0.79 TDP1 (0.45) CCNE1CDK2CDK5CHRNA7
SCHEMBL11252606 0.78 TDP1 (0.44) CCNE1CDK2CDK5CHRNA7
SCHEMBL11267468 0.77 ANPEP (0.38) DGAT2KLKB1CYP3A4ANPEP
SCHEMBL11267832 0.77 TDP1 (0.45) CCNE1CDK2CDK5CHRNA7
SCHEMBL11259018 0.76 ALDH1A1 (0.39) KLKB1ANPEP
SCHEMBL11261376 0.76 KDM4E (0.41) CDK5NPC1RAB9ACHRNA7
SCHEMBL11260207 0.75 TDP1 (0.35) CDK5CHRNA7
SCHEMBL11266460 0.75 CDK5 (0.38) CCNE1CDK2CDK5CHRNA7
SCHEMBL11263036 0.74 ALDH1A1 (0.40) DGAT2KLKB1ANPEP
SCHEMBL11260439 0.74 TDP1 (0.47) CCNE1CDK2CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed