SCHEMBL11260439

SCHEMBL11260439

O=C(O)Cc1cccc2c(C3CC3)nccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.47
CYP1A2 P05177 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
AKR1B1 P15121 1/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.37
SLC22A12 Q96S37 3/20 0.37
CDK2 P24941 2/20 0.36
CXCL8 P10145 2/20 0.36
CCNA2 P20248 1/20 0.36
CCNA1 P78396 1/20 0.36
GLA P06280 1/20 0.36
STING1 Q86WV6 1/20 0.36
PPARG P37231 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
CCNE1 P24864 1/20 0.35
CDK5 Q00535 1/20 0.35
PTGS2 P35354 2/20 0.35
AKR1B10 O60218 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11267832 0.94 TDP1 (0.45) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11269174 0.94 TDP1 (0.45) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11252606 0.93 TDP1 (0.44) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11266460 0.81 CDK5 (0.38) TDP1KDM4ECDK2GLACCNE1
SCHEMBL19099076 0.80 KDM4E (0.56) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL4194024 0.77 TDP1 (0.54) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL11261376 0.77 KDM4E (0.41) TDP1KDM4EMAPTCDK5
SCHEMBL11263232 0.76 PKM (0.40) TDP1KDM4EMAPT
SCHEMBL11311256 0.76 TDP1 (0.53) TDP1CYP1A2KDM4EMAPTAKR1B1
SCHEMBL69234 0.76 TDP1 (0.76) TDP1CYP1A2KDM4EMAPTAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed