SCHEMBL11246607

SCHEMBL11246607

CCCCOC(=O)c1ccc2nc(N)[nH]c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.55
LMNA P02545 3/20 0.55
TSHR P16473 3/20 0.55
CYP2C19 P33261 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2C9 P11712 1/20 0.55
PDE4D Q08499 1/20 0.55
MAPT P10636 3/20 0.54
GAA P10253 2/20 0.54
PKM P14618 1/20 0.54
ABL1 P00519 1/20 0.52
FABP6 P51161 1/20 0.52
PKN1 Q16512 1/20 0.50
PKN2 Q16513 1/20 0.50
SIRT2 Q8IXJ6 3/20 0.49
SIRT1 Q96EB6 2/20 0.49
SIRT3 Q9NTG7 1/20 0.49
ESR1 P03372 4/20 0.49
CYP2D6 P10635 3/20 0.49
NPC1 O15118 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11246587 0.90 CYP1A2 (0.55) CYP1A2LMNATSHRCYP2C19CYP3A4
SCHEMBL8283877 0.87 PKN1 (0.64) CYP1A2LMNACYP3A4MAPTABL1
SCHEMBL9306377 0.85 PKN1 (0.50) CYP1A2LMNATSHRCYP2C19CYP3A4
SCHEMBL4682076 0.80 ALDH1A1 (0.64) LMNACYP2C9MAPTGAAPKM
SCHEMBL19118043 0.79 TSHR (0.49) CYP1A2LMNATSHRCYP2C19CYP3A4
SCHEMBL11540940 0.78 FABP6 (0.58) ABL1FABP6RAB9AALDH1A1SMN1; SMN2
SCHEMBL14046197 0.77 CYP1A2 (0.57) CYP1A2LMNATSHRCYP2C19CYP3A4
SCHEMBL9178141 0.77 LMNA (0.52) CYP1A2LMNATSHRCYP2C19CYP3A4
SCHEMBL31317898 0.77 LMNA (0.52) CYP1A2LMNATSHRCYP2C19CYP3A4
SCHEMBL11148656 0.76 HCRTR1 (0.53) CYP1A2LMNACYP3A4MAPTPKN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4316021-A VIRICIDES ELI LILLY AND COMPANY (US) 1982-02-16 US disclosed
US-4243813-A VIRICIDES ELI LILLY AND COMPANY (US) 1981-01-06 US disclosed
US-4196125-A VIRICIDES ELI LILLY AND COMPANY (US) 1980-04-01 US disclosed
US-4118573-A ANTIVIRAL AGENTS ELI LILLY AND COMPANY (US) 1978-10-03 US disclosed
US-4018790-A VIRICIDES ELI LILLY AND COMPANY (US) 1977-04-19 US disclosed