SCHEMBL11247740

SCHEMBL11247740

CCCCCc1nc(NN)ccc1-c1ccncc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
DHFR P00374 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
GSK3B P49841 2/20 0.35
NPC1 O15118 1/20 0.35
NFKB1 P19838 1/20 0.35
S1PR1 P21453 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LATS1 O95835 3/20 0.35
LATS2 Q9NRM7 3/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11074069 0.82 GABRP (0.47) CYP3A4CYP2D6DHFRSMN1; SMN2ALDH1A1
SCHEMBL11255710 0.79 AAK1 (0.37) CYP3A4GSK3BS1PR1PDE3BPDE3A
SCHEMBL11176428 0.79 CYP3A4 (0.39) CYP3A4CYP2D6DHFRSMN1; SMN2ALDH1A1
SCHEMBL11071690 0.79 ADORA2B (0.42) ALDH1A1ADORA2BNAAAADORA2AADORA1
SCHEMBL11164012 0.77 GABRP (0.51) CYP3A4CYP2D6DHFRSMN1; SMN2ALDH1A1
SCHEMBL11247476 0.77 PDE3B (0.36) CYP3A4CYP2D6DHFRSMN1; SMN2ALDH1A1
SCHEMBL7272491 0.75 DYRK1A (0.47) CYP3A4CYP2D6SMN1; SMN2ALDH1A1MAPT
SCHEMBL11063569 0.74 PDE3B (0.42) ALDH1A1MAPTPDE3BPDE3AADORA2B
SCHEMBL11069278 0.74 ADORA2B (0.43) GSK3BADORA2BADORA2AADORA1
SCHEMBL7280225 0.74 MAPT (0.40) CYP3A4CYP2D6SMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4351941-A Pyridinyl-pyridines STERLING DRUG INC. (US) 1982-09-28 US disclosed
US-4331672-A 5-(Pyridinyl)pyridine-2-hydrazines, their preparation and their cardiotonic use STERLING DRUG INC. (US) 1982-05-25 US disclosed