SCHEMBL11247894

SCHEMBL11247894

O=C(O)C(Br)c1c(Cl)cccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
AKR1B1 P15121 1/20 0.42
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 2/20 0.40
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
MEN1 O00255 1/20 0.40
FEN1 P39748 2/20 0.37
CXCL8 P10145 1/20 0.37
SLC1A3 P43003 1/20 0.37
SLC1A2 P43004 1/20 0.37
CACNA2D1 P54289 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNB1 Q02641 1/20 0.35
ERCC5 P28715 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28852475 0.87 CES2 (0.41) TSHRAKR1B1ALDH1A1CES2CES1
SCHEMBL11241971 0.83 ALDH1A1 (0.41) TSHRAKR1B1ALDH1A1KMT2ACES2
SCHEMBL5179498 0.81 ALDH1A1 (0.40) TSHRAKR1B1ALDH1A1KMT2ACES2
SCHEMBL11271848 0.80 ALDH1A1 (0.45) TSHRAKR1B1ALDH1A1KMT2ACES2
SCHEMBL365284 0.77 MEN1 (0.46) ALDH1A1KMT2ACES2CES1MEN1
SCHEMBL5112227 0.77 MEN1 (0.46) ALDH1A1KMT2ACES2CES1MEN1
SCHEMBL8128086 0.77 MEN1 (0.46) ALDH1A1KMT2ACES2CES1MEN1
SCHEMBL9274763 0.76 PDK1 (0.39) ALDH1A1KMT2AMEN1
SCHEMBL9125705 0.76 KMT2A (0.40) TSHRALDH1A1KMT2AMEN1
SCHEMBL11686588 0.74 KMT2A (0.47) TSHRAKR1B1ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4318915-A Substituted guandines and methods of preparation thereof BEIERSDORF AKTIENGESELLSCHAFT (DE) 1982-03-09 US disclosed