SCHEMBL11248331

SCHEMBL11248331

N#CCc1ccsc1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
TP53 P04637 1/20 0.49
ALOX15 P16050 1/20 0.49
MAPK1 P28482 1/20 0.49
LMNA P02545 1/20 0.37
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
PTGS2 P35354 1/20 0.35
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
GRM6 O15303 1/20 0.33
PDPK1 O15530 1/20 0.33
PTGS1 P23219 1/20 0.33
CYP2A6 P11509 1/20 0.33
PTPRC P08575 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
ATR Q13535 1/20 0.32
CYP1A1 P04798 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5111011 0.75 TP53 (0.57) KMT2ATP53ALOX15MAPK1ALDH1A1
SCHEMBL7386191 0.75 KMT2A (0.53) KMT2ATP53ALOX15MAPK1ALDH1A1
SCHEMBL27659211 0.75 TP53 (0.53) KMT2ATP53ALOX15MAPK1ALDH1A1
SCHEMBL6064370 0.72 GRM6 (0.44) KMT2ATP53ALOX15MAPK1LMNA
SCHEMBL1408548 0.72 TP53 (0.54) KMT2ATP53ALOX15MAPK1ALDH1A1
SCHEMBL901920 0.72 KMT2A (0.50) KMT2ATP53ALOX15MAPK1ALDH1A1
SCHEMBL27942120 0.70 TP53 (0.49) KMT2ATP53ALOX15MAPK1HPGD
SCHEMBL1520751 0.70 KMT2A (0.71) KMT2ATP53ALOX15MAPK1LMNA
SCHEMBL1343377 0.70 DPP4 (0.56) KMT2AMAPK1LMNAALDH1A1HPGD
SCHEMBL3676147 0.70 CYP2A6 (0.37) ALDH1A1HPGDCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0013424-B1 SPIRO(DIBENZO(B,F)THIEPINE-PIPERIDINES), INTERMEDIATE PRODUCTS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1982-11-17 EP disclosed
EP-0013424-A1 Spiro(dibenzo(b,f)thiepine-piperidines), intermediate products for their preparation and medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1980-07-23 EP disclosed
US-4198420-A Spiro[dibenz(b,f)thiepin-piperidine]s AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed
US-4198419-A Phenylthiophenylpiperidines AMERICAN HOECHST CORPORATION (US) 1980-04-15 US disclosed