SCHEMBL11248371

SCHEMBL11248371

CNc1ncc(-c2cccnc2)cc1C#N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.47
CYP11B2 P19099 2/20 0.46
ADORA1 P30542 1/20 0.45
EPHX2 P34913 1/20 0.44
PRMT6 Q96LA8 1/20 0.44
CYP17A1 P05093 1/20 0.43
CYP11B1 P15538 1/20 0.43
ALDH1A1 P00352 5/20 0.43
CYP2A6 P11509 4/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CYP3A4 P08684 3/20 0.43
CYP1A2 P05177 2/20 0.43
NEK1 Q96PY6 1/20 0.42
PDGFRB P09619 2/20 0.41
PDGFRA P16234 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11247724 0.84 PIK3CD (0.44) CHEK1ADORA1ALDH1A1NPSR1TDP1
SCHEMBL27241764 0.83 KDR (0.45) CHEK1CYP11B2CYP17A1CYP11B1ALDH1A1
SCHEMBL10841297 0.79 ALDH1A1 (0.45) CYP11B2ADORA1EPHX2PRMT6CYP17A1
SCHEMBL7279694 0.78 PDGFRB (0.51) CHEK1CYP11B2CYP17A1CYP11B1ALDH1A1
SCHEMBL11248859 0.78 ALDH1A1 (0.41) CYP11B2CYP11B1ALDH1A1NPSR1TDP1
SCHEMBL7282308 0.78 ALDH1A1 (0.71) CHEK1CYP11B2CYP17A1CYP11B1ALDH1A1
SCHEMBL27241705 0.77 KDR (0.41) CHEK1CYP11B2CYP17A1CYP11B1ALDH1A1
SCHEMBL7285793 0.77 CHEK1 (0.47) CHEK1ALDH1A1CYP2A6NPSR1TDP1
SCHEMBL11242985 0.75 CCNC (0.52) CYP11B2ALDH1A1TDP1CYP3A4CYP1A2
SCHEMBL11240500 0.75 KDM4E (0.39) CYP11B2CYP11B1ALDH1A1NPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362734-A 2-(Substituted-amino)-5-(pyridinyl-nicotinonitriles, and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed