SCHEMBL11248859

SCHEMBL11248859

CNc1ncc(-c2cccnc2C)cc1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
GRM5 P41594 2/20 0.40
CYP11B2 P19099 2/20 0.39
CYP11B1 P15538 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.37
KDM4E B2RXH2 3/20 0.37
GAA P10253 1/20 0.37
ALOX5AP P20292 1/20 0.37
FEN1 P39748 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
HPGD P15428 3/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11227756 0.81 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4CYP11B2CYP11B1
SCHEMBL10843843 0.78 ALDH1A1 (0.38) ALDH1A1CYP1A2CYP3A4MAPK1HSD17B10
SCHEMBL11248371 0.78 CHEK1 (0.47) ALDH1A1CYP1A2CYP3A4HSD17B10CLK4
SCHEMBL7285793 0.78 CHEK1 (0.47) ALDH1A1CYP1A2CYP3A4MAPK1HSD17B10
SCHEMBL11247724 0.76 PIK3CD (0.44) ALDH1A1CYP1A2CYP3A4CLK4KDM4E
SCHEMBL15730158 0.74 CYP11B2 (0.52) CYP11B2CYP11B1ALOX5APFEN1MKNK1
SCHEMBL11242985 0.73 CCNC (0.52) ALDH1A1CYP1A2CYP3A4MAPK1HSD17B10
SCHEMBL11240500 0.73 KDM4E (0.39) ALDH1A1CYP1A2CYP3A4MAPK1HSD17B10
SCHEMBL31023872 0.72 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4MAPK1HSD17B10
SCHEMBL3390876 0.72 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4MAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362734-A 2-(Substituted-amino)-5-(pyridinyl-nicotinonitriles, and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed