SCHEMBL11242985

SCHEMBL11242985

CCc1cnccc1-c1cnc(NC)c(C#N)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.52
CDK8 P49336 1/20 0.52
PDE3B Q13370 3/20 0.38
PDE3A Q14432 3/20 0.38
AAK1 Q2M2I8 1/20 0.37
LRRK2 Q5S007 2/20 0.37
ALDH1A1 P00352 4/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
HSD17B10 Q99714 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
MAPK1 P28482 1/20 0.36
PDE10A Q9Y233 1/20 0.36
KDM4E B2RXH2 3/20 0.35
CYP2C19 P33261 3/20 0.35
LMNA P02545 2/20 0.35
HPGD P15428 2/20 0.35
XIAP P98170 1/20 0.35
BIRC2 Q13490 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11237350 0.82 CCNC (0.54) CCNCCDK8PDE3BPDE3AAAK1
SCHEMBL10844104 0.80 CCNC (0.46) CCNCCDK8PDE3BPDE3ALRRK2
SCHEMBL11247724 0.78 PIK3CD (0.44) CCNCCDK8PDE3BPDE3ALRRK2
SCHEMBL11160803 0.77 SIRT3 (0.41) CCNCCDK8ALDH1A1PDE10AKDM4E
SCHEMBL11248371 0.75 CHEK1 (0.47) ALDH1A1CYP1A2CYP3A4HSD17B10CLK4
SCHEMBL11450302 0.73 CCNC (0.70) CCNCCDK8PDE3BPDE3ALRRK2
SCHEMBL11248859 0.73 ALDH1A1 (0.41) ALDH1A1CYP1A2CYP3A4HSD17B10CLK4
SCHEMBL11238008 0.70 GSK3A (0.45) CDK8PDE3BPDE3ALRRK2ALDH1A1
SCHEMBL4544610 0.70 CCNC (0.49) CCNCCDK8PDE3BPDE3AALDH1A1
SCHEMBL7285793 0.69 CHEK1 (0.47) ALDH1A1CYP1A2CYP3A4HSD17B10CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4362734-A 2-(Substituted-amino)-5-(pyridinyl-nicotinonitriles, and their cardiotonic use STERLING DRUG INC. (US) 1982-12-07 US disclosed