SCHEMBL11248787

SCHEMBL11248787

O=C=Nc1nccc(Cl)n1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
TRPA1 O75762 1/20 0.32
TAAR1 Q96RJ0 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27545997 0.76 ALOX15 (0.39) MAPK1TDP1TRPA1GABRA1GABRB2
SCHEMBL9661250 0.74 MAPK1 (0.39) MAPK1TDP1GABRA1GABRB2
SCHEMBL3050642 0.71
SCHEMBL11193798 0.69 MAPK1 (0.31) MAPK1TDP1
SCHEMBL11038525 0.69 MAPK8 (0.36) TAAR1GABRA1GABRB2
SCHEMBL713341 0.69 CYP3A4 (0.30)
SCHEMBL17059628 0.68 MAPK1 (0.34) MAPK1TDP1GABRA1GABRB2
SCHEMBL10806196 0.68 MAPK1 (0.34) MAPK1TDP1
SCHEMBL10547105 0.68 MAPK1 (0.34) MAPK1TDP1
SCHEMBL1191366 0.68 TRPA1 (0.56) MAPK1TDP1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106810512-B IDH2 mutant inhibitor and application thereof 江苏省中医药研究院 2019-09-10 CN disclosed
CN-106810512-A IDH2 mutant inhibitor and application thereof 江苏省中医药研究院 2017-06-09 CN disclosed
EP-0044209-A1 Herbicidal sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-01-20 EP disclosed