SCHEMBL11248816

SCHEMBL11248816

COc1ccccc1C1=NCC2CN(C)CCN2c2ccc(Cl)cc21

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HRH4 Q9H3N8 1/20 0.41
HTR2A P28223 3/20 0.41
HTR2C P28335 2/20 0.41
HTR1A P08908 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
HTR1E P28566 1/20 0.41
HTR7 P34969 1/20 0.41
HTR2B P41595 1/20 0.41
HTR3A P46098 1/20 0.41
HTR5A P47898 1/20 0.41
OPRK1 P41145 4/20 0.39
PDE4D Q08499 4/20 0.39
ADRA1A P35348 2/20 0.39
NR1I2 O75469 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
PTGS2 P35354 1/20 0.39
CHRNA4 P43681 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11266201 0.89 OPRK1 (0.47) SMN1; SMN2HTR2AHTR2COPRK1PDE4D
Hydrochloric Acid SCHEMBL11431914 0.83 OPRK1 (0.56) HPGDHTR2COPRK1PDE4DADRA1A
SCHEMBL10858544 0.78 OPRK1 (0.38) HRH4HTR2AHTR2CHTR1AHTR7
SCHEMBL11266170 0.73 HPGD (0.51) HPGDSMN1; SMN2HTR2AHTR2CHTR1A
SCHEMBL11251836 0.73 OPRK1 (0.49) HPGDHTR2COPRK1PDE4DADRA1A
Hydrochloric Acid SCHEMBL11251814 0.73 EBP (0.43) HTR2COPRK1PDE4DADRA1ANR1I2
Hydrochloric Acid SCHEMBL11255176 0.72 OPRK1 (0.40) HTR2AHTR2CHTR2BOPRK1PDE4D
SCHEMBL9652997 0.72 CCKBR (0.46) HTR2AHTR2CHTR1AHTR1DHTR7
Hydrochloric Acid SCHEMBL11248904 0.71 OPRK1 (0.40) HPGDHTR2AHTR2CHTR2BOPRK1
SCHEMBL11261476 0.70 OPRK1 (0.45) SMN1; SMN2HTR2AHTR2COPRK1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4338314-A [1,2]Anellated-7-phenyl-1,4-benzodiazepine and pharmaceutical compositions thereof and use for treatment of ulcers KALI-CHEMIE PHARMA GMBH (DE) 1982-07-06 US disclosed