SCHEMBL11266201

SCHEMBL11266201

CN1CCN2c3ccc(Cl)cc3C(c3ccccc3Cl)=NCC2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 4/20 0.47
PDE4D Q08499 4/20 0.47
GABRA1 P14867 4/20 0.47
GABRA5 P31644 4/20 0.47
GABRA2 P47869 4/20 0.47
GABRG2 P18507 3/20 0.47
GABRB3 P28472 3/20 0.47
GABRA3 P34903 3/20 0.47
ADRA1A P35348 2/20 0.47
HTR2A P28223 1/20 0.47
CHRM2 P08172 1/20 0.46
ADRA2A P08913 1/20 0.46
NR1I2 O75469 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
HTR2C P28335 1/20 0.45
PTGS2 P35354 1/20 0.45
CHRNA4 P43681 1/20 0.45
SLC6A3 Q01959 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
TP53 P04637 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11248816 0.89 HPGD (0.51) OPRK1PDE4DGABRA1GABRA5GABRA2
Hydrochloric Acid SCHEMBL11431914 0.87 OPRK1 (0.56) OPRK1PDE4DGABRA1GABRA5GABRA2
SCHEMBL10858544 0.82 OPRK1 (0.38) OPRK1PDE4DGABRA1GABRA5GABRA2
SCHEMBL11261476 0.80 OPRK1 (0.45) OPRK1PDE4DGABRA1GABRA5GABRA2
SCHEMBL10919992 0.77 OPRK1 (0.51) OPRK1PDE4DGABRA1GABRA5GABRA2
SCHEMBL10919997 0.77 OPRK1 (0.51) OPRK1PDE4DGABRA1GABRA5GABRA2
SCHEMBL7313742 0.77 OPRK1 (0.54) OPRK1PDE4DGABRA1GABRA5GABRA2
Hydrochloric Acid SCHEMBL7348131 0.76 GABRA1 (0.50) OPRK1PDE4DGABRA1GABRA5GABRA2
SCHEMBL10918118 0.76 OPRK1 (0.54) OPRK1PDE4DGABRA1GABRA5GABRA2
SCHEMBL10918115 0.76 OPRK1 (0.54) OPRK1PDE4DGABRA1GABRA5GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4338314-A [1,2]Anellated-7-phenyl-1,4-benzodiazepine and pharmaceutical compositions thereof and use for treatment of ulcers KALI-CHEMIE PHARMA GMBH (DE) 1982-07-06 US disclosed