SCHEMBL11250351

SCHEMBL11250351

CCCCCCCCCCCCCCCCNc1ccc(C(=O)CC(=O)O)cc1F

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 3/20 0.49
PLK1 P53350 3/20 0.46
EPHX2 P34913 1/20 0.43
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
RARB P10826 1/20 0.41
S1PR3 Q99500 1/20 0.41
NAAA Q02083 1/20 0.40
XDH P47989 1/20 0.40
HAO1 Q9UJM8 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11258895 0.90 HCAR3 (0.47) HCAR3PLK1EPHX2THRATHRB
SCHEMBL11255414 0.88 HCAR3 (0.62) HCAR3PLK1EPHX2THRBRARB
SCHEMBL15412525 0.88 HCAR3 (0.62) HCAR3PLK1EPHX2THRBRARB
SCHEMBL11262794 0.86 HCAR3 (0.61) HCAR3PLK1EPHX2THRBRARB
SCHEMBL11270514 0.85 PLK1 (0.43) HCAR3PLK1EPHX2THRATHRB
SCHEMBL11258316 0.85 HCAR3 (0.49) HCAR3PLK1EPHX2RARBNAAA
SCHEMBL11262791 0.83 HCAR3 (0.50) HCAR3PLK1EPHX2RARBNAAA
Hydrochloric Acid SCHEMBL11250653 0.83 HCAR3 (0.47) HCAR3PLK1EPHX2RARBCNR2
SCHEMBL11258578 0.83 MAPT (0.55) HCAR3PLK1EPHX2
SCHEMBL11260606 0.83 ALDH1A1 (0.50) HCAR3PLK1EPHX2THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4333940-A Ring-fluorinated 4-(monosubstituted-amino) phenyl compounds in inhibiting atherosclerotic lesion development AMERICAN CYANAMID COMPANY (US) 1982-06-08 US disclosed
US-4243609-A ANTILIPEMIC AGENTS, ANTIATHEROSCLEROTIC AGENTS AMERICAN CYANAMID COMPANY (US) 1981-01-06 US disclosed
EP-0003663-A2 Amino-substituted phenyl and heteroaryl compounds, process for their preparation and pharmaceutical compositions containing them AMERICAN CYANAMID COMPANY (US) 1979-08-22 EP disclosed