SCHEMBL11255165

SCHEMBL11255165

CN(C)c1ccc(-c2nccc3c(CC(N)=O)cccc23)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.38
MAP2K7 O14733 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
PARP1 P09874 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
SYK P43405 3/20 0.35
APP P05067 1/20 0.35
ADK P55263 1/20 0.35
HSP90AA1 P07900 1/20 0.35
AOC3 Q16853 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11250186 0.89 PTGDR2 (0.43) CNR2ROCK2ROCK1OPRM1OPRD1
SCHEMBL11261717 0.84 NPSR1 (0.44) HTR2BNPSR1MAPTPTGDR2ALDH1A1
SCHEMBL11257859 0.84 JAK2 (0.41) NPSR1TP53GAAMAPTALDH1A1
SCHEMBL11248945 0.84 IDO1 (0.42) PTGDR2ALDH1A1HTT
SCHEMBL11254978 0.78 SYK (0.35) TP53GAAMAPTSYKADK
SCHEMBL11257961 0.77 KDM4E (0.42) TP53MAPTPTGDR2ALDH1A1
SCHEMBL11246786 0.74 LMNA (0.48) NPSR1GAAMAPTPTGDR2ALDH1A1
SCHEMBL11251835 0.73 TDP1 (0.54) HTR2BMAPTPTGDR2ALDH1A1
SCHEMBL11257643 0.73 PSEN1 (0.39) CNR2ROCK2ROCK1HTR2CHTR2B
SCHEMBL11262913 0.73 ALDH1A1 (0.39) CNR2ROCK2ROCK1HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed