SCHEMBL11248945

SCHEMBL11248945

NC(=O)Cc1cccc2c(-c3ccc(Cl)cc3)nccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
CSNK2A2 P19784 2/20 0.41
CSNK2B P67870 2/20 0.41
PTGDR2 Q9Y5Y4 2/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
KDR P35968 1/20 0.39
CYP2C19 P33261 1/20 0.38
NPY5R Q15761 1/20 0.38
MAP4K4 O95819 2/20 0.37
PDE10A Q9Y233 1/20 0.37
KDM4E B2RXH2 1/20 0.36
DRD2 P14416 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HTT P42858 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11255704 0.88 PTGDR2 (0.49) IDO1TDO2CSNK2A2CSNK2BPTGDR2
SCHEMBL11261717 0.88 NPSR1 (0.44) TDO2PTGDR2PDE3BPDE3AKDM4E
SCHEMBL11255165 0.84 CNR2 (0.38) PTGDR2ALDH1A1HTT
SCHEMBL11266566 0.84 KDR (0.40) IDO1TDO2CSNK2A2CSNK2BPTGDR2
SCHEMBL11500393 0.83 PTGDR2 (0.45) IDO1TDO2CSNK2A2CSNK2BPTGDR2
SCHEMBL11262405 0.80 TDO2 (0.48) IDO1TDO2CSNK2A2CSNK2BPTGDR2
SCHEMBL11253962 0.80 TDO2 (0.45) IDO1TDO2CSNK2A2CSNK2BPTGDR2
SCHEMBL11256404 0.79 TDO2 (0.47) IDO1TDO2CSNK2A2CSNK2BPTGDR2
SCHEMBL11251835 0.76 TDP1 (0.54) TDO2PTGDR2PDE3BPDE3AKDM4E
SCHEMBL11248931 0.76 TDO2 (0.44) IDO1TDO2CSNK2A2CSNK2BPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337256-A ANTIINFLAMMATORY AGENTS; ANTIAGGLOMERANTS; ENZYME INHIBITORS; ANTIULCER AGENTS TEIKOKU HORMONE MANUFACTURING CO., LTD. (JP) 1982-06-29 US disclosed
EP-0013411-A1 Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them TEIKOKU HORMONE MFG. CO., LTD. (JP) 1980-07-23 EP disclosed