SCHEMBL11256205

SCHEMBL11256205

COC(=O)NC(c1ccccc1)C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.53
GABRB1 P18505 1/20 0.46
GABRB2 P47870 1/20 0.46
KMT2A Q03164 3/20 0.46
TACR3 P29371 1/20 0.45
MEN1 O00255 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
GAA P10253 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
PRCP P42785 1/20 0.44
CTSL P07711 4/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
MAPT P10636 1/20 0.43
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15045485 0.84 HTT (0.54) HTTGABRB1GABRB2KMT2AMEN1
SCHEMBL13132826 0.84 HTT (0.54) HTTGABRB1GABRB2KMT2AMEN1
SCHEMBL17777055 0.82 TACR3 (0.47) HTTKMT2ATACR3MEN1PRCP
SCHEMBL16989173 0.82 TACR3 (0.49) HTTKMT2ATACR3MEN1PRCP
SCHEMBL16989172 0.82 TACR3 (0.49) HTTKMT2ATACR3MEN1PRCP
SCHEMBL250886 0.82 TACR3 (0.49) HTTKMT2ATACR3MEN1PRCP
SCHEMBL12965965 0.80 HTT (0.54) HTTGABRB1GABRB2KMT2AMEN1
SCHEMBL10338251 0.79 GAA (0.50) HTTKMT2ATACR3MEN1GAA
SCHEMBL8689297 0.78 LMNA (0.49) KMT2ATACR3MEN1PRCPCTSL
SCHEMBL29972950 0.76 CYP1A2 (0.43) HTTGABRB1GABRB2KMT2ATACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4315020-A Oxazoline (trifluoroethyl) amine SCIENCE UNION ET CIE (FR) 1982-02-09 US disclosed
US-4315019-A Novel aryltrifluoroethylamines and processes for producing the same SCIENCE UNION ET CIE (FR) 1982-02-09 US disclosed
US-4267345-A 2-//PYRROL-2-YL, THIEN-2-YL, OR FUR-2-YL/-ALPHA-TRIFLUOROALKYL-AMINOOXAZOLINES; HYPOTENSIVE AGENTS SCIENCE UNION ET CIE (FR) 1981-05-12 US disclosed