SCHEMBL11257889

SCHEMBL11257889

C[C@]12CCC(=O)C(C(=O)c3ccccc3)[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 4/20 0.53
CYP19A1 P11511 11/20 0.52
AKR1B10 O60218 1/20 0.48
AKR1B1 P15121 1/20 0.48
OR51E2 Q9H255 1/20 0.48
GPBAR1 Q8TDU6 3/20 0.46
SHBG P04278 2/20 0.46
SERPINA6 P08185 2/20 0.46
LMNA P02545 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPK1 P28482 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11257890 1.00 HSD17B3 (0.53) HSD17B3CYP19A1AKR1B10AKR1B1OR51E2
SCHEMBL11235253 0.85 CYP19A1 (0.51) CYP19A1OR51E2GPBAR1SHBGSERPINA6
SCHEMBL11235256 0.85 CYP19A1 (0.51) CYP19A1OR51E2GPBAR1SHBGSERPINA6
SCHEMBL11239863 0.83 SRD5A1 (0.43) AKR1B10AKR1B1GPBAR1
SCHEMBL11239844 0.83 SRD5A1 (0.43) AKR1B10AKR1B1GPBAR1
SCHEMBL10185940 0.81 CYP19A1 (0.55) HSD17B3CYP19A1AKR1B10AKR1B1OR51E2
SCHEMBL11242981 0.79 CYP17A1 (0.50) GPBAR1
SCHEMBL11242975 0.79 CYP17A1 (0.50) GPBAR1
SCHEMBL11243490 0.79 SRD5A2 (0.59) AKR1B10AKR1B1GPBAR1LMNAMEN1
SCHEMBL11243498 0.79 SRD5A2 (0.59) AKR1B10AKR1B1GPBAR1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4317817-A SKIN DISORDERS; ACEME; ENZYME INHIBITORS RICHARDSON-MERRELL INC. (US) 1982-03-02 US disclosed