SCHEMBL11258489

SCHEMBL11258489

COc1cc2c(c(Br)c1OC)CCCCN2c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 2/20 0.41
TSHR P16473 1/20 0.41
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
LMNA P02545 2/20 0.38
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
CYP1A2 P05177 1/20 0.35
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7620197 0.76 DRD1 (0.45) ALDH1A1KDM4ETSHRMEN1KMT2A
Hydrochloric Acid SCHEMBL11252603 0.75 KDM4E (0.41) ALDH1A1MAPTKDM4ETSHRMEN1
SCHEMBL11343586 0.72 MAPT (0.43) ALDH1A1MAPTKDM4ETSHRMEN1
SCHEMBL10655982 0.68 CYP1A1 (0.38) ALDH1A1MAPTTSHRKMT2ALMNA
SCHEMBL7629632 0.67 TUBB4A (0.50) TSHRTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL7621171 0.63 MAOB (0.53) MAPTKDM4EMEN1KMT2ALMNA
SCHEMBL7618224 0.63 HDAC1 (0.45) ALDH1A1MAPTKDM4EMEN1KMT2A
Bromide SCHEMBL11460380 0.62 POLB (0.35) KDM4ELMNAHTT
SCHEMBL13928826 0.62 MAOA (0.51) ALDH1A1MAPTKDM4ETSHRMEN1
SCHEMBL27757915 0.62 DRD1 (0.52) ALDH1A1KDM4ETSHRTUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4359464-A 3-Furylmethyl-6-halo-7,8-dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepines and antihypertensive use thereof SMITHKLINE BECKMAN CORPORATION (US) 1982-11-16 US disclosed
US-4352754-A HYPOTENSIVE, ANTI-PARKINSON SMITHKLINE CORPORATION (US) 1982-10-05 US disclosed
US-4255422-A DIURETICS, TREATMENT OF CARDIOVASCULAR DISORDERS SMITHKLINE CORPORATION (US) 1981-03-10 US disclosed
US-4160765-A Method for 6-bromination of 1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine compounds SMITHKLINE CORPORATION (US) 1979-07-10 US disclosed