SCHEMBL11258667

SCHEMBL11258667

N#CNc1nc2c(C(=O)c3cccs3)cccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.44
RAB9A P51151 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 3/20 0.42
ALOX15 P16050 1/20 0.42
MAPT P10636 3/20 0.40
ABL1 P00519 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 2/20 0.40
NFKB1 P19838 2/20 0.40
GMNN O75496 1/20 0.40
TUBB4A P04350 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAOA P21397 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11258510 0.81 ABL1 (0.62) NPC1RAB9ASMN1; SMN2KDM4ELMNA
SCHEMBL11258664 0.76 NPC1 (0.58) NPC1RAB9ASMN1; SMN2KDM4ELMNA
SCHEMBL11258670 0.75 ABL1 (0.69) NPC1RAB9ASMN1; SMN2KDM4ELMNA
SCHEMBL27868475 0.70 LMNA (0.49) NPC1RAB9ASMN1; SMN2KDM4ELMNA
SCHEMBL11782292 0.68 MGAM (0.46) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1
SCHEMBL9148337 0.66 LMNA (0.85) NPC1RAB9ASMN1; SMN2LMNAALOX15
SCHEMBL29152812 0.65 ALOX15 (0.49) NPC1RAB9ASMN1; SMN2KDM4ELMNA
SCHEMBL6841863 0.64 RIPK1 (0.48) RIPK1PARP1PKN1PKN2PLK4
SCHEMBL11705968 0.63 CYP2C9 (0.47) NPC1RAB9AKDM4ELMNAALOX15
SCHEMBL11195206 0.63 ALOX15 (0.62) NPC1RAB9ASMN1; SMN2LMNAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4321393-A Method for preparing 2-cyanamidobenzimidazoles or 2-cyanamidobenzoxazoles SMITHKLINE CORPORATION (US) 1982-03-23 US disclosed
US-4285878-A N-Phenyl-N'-cyano-O-phenylisoureas SMITHKLINE CORPORATION (US) 1981-08-25 US disclosed