SCHEMBL11259609

SCHEMBL11259609

COc1ccc(C(C)(C)C)cc1C(O)(c1ccccc1)C(C)N1CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
HTT P42858 4/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KCNA5 P22460 2/20 0.36
ALDH1A1 P00352 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LPAR5 Q9H1C0 1/20 0.36
NPY2R P49146 1/20 0.36
KCNH2 Q12809 1/20 0.36
NPSR1 Q6W5P4 2/20 0.36
RAB9A P51151 2/20 0.36
LMNA P02545 1/20 0.36
NR3C2 P08235 1/20 0.36
NPC1 O15118 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 1/20 0.36
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11260709 0.83 KCNA5 (0.36) MEN1KMT2AHTTCYP3A4CYP2D6
SCHEMBL11253547 0.82 HTT (0.36) MEN1KMT2AHTTCYP3A4CYP2D6
SCHEMBL11264980 0.79 MEN1 (0.41) MEN1KMT2AHTTCYP3A4CYP2D6
SCHEMBL11259393 0.78 ALDH1A1 (0.37) ALDH1A1SMN1; SMN2NPSR1RAB9AL3MBTL1
SCHEMBL364905 0.78 KCNA5 (0.50) CYP3A4CYP2D6CYP2C19KCNA5ALDH1A1
SCHEMBL11268090 0.73 GLRA1 (0.39) MEN1KMT2AALDH1A1SMN1; SMN2RAB9A
SCHEMBL11258069 0.72 KCNA5 (0.39) MEN1KMT2ACYP3A4CYP2D6CYP2C19
SCHEMBL11257390 0.72 MEN1 (0.34) MEN1KMT2AHTTCYP3A4CYP2D6
SCHEMBL12890839 0.71 KCNA5 (0.52) CYP3A4CYP2D6CYP2C19KCNA5ALDH1A1
SCHEMBL11251766 0.70 P4HB (0.36) MEN1KMT2AHTTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4361573-A α,α-Diaryl-β-(tert-amino)-propanols and diuretic pharmaceutical compositions containing them TEMMLER AG (CH) 1982-11-30 US disclosed
US-4025633-A DIURETICS, SALURETICS FIRMA TEMMLER A.G. (CH) 1977-05-24 US disclosed