SCHEMBL11259683

SCHEMBL11259683

COC(=O)COc1cccc(/C=C(\C)[N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYSLTR2 Q9NS75 1/20 0.49
CYSLTR1 Q9Y271 1/20 0.49
PTGS2 P35354 1/20 0.49
FBP1 P09467 1/20 0.49
POLB P06746 1/20 0.47
ABL1 P00519 1/20 0.45
EGFR P00533 1/20 0.45
ABL2 P42684 1/20 0.45
ALDH1A1 P00352 4/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
S1PR4 O95977 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
S1PR1 P21453 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11259689 1.00 CYSLTR2 (0.49) CYSLTR2CYSLTR1PTGS2FBP1POLB
SCHEMBL11246287 0.84 PTGS2 (0.64) PTGS2FBP1ABL1EGFRABL2
SCHEMBL11246288 0.84 PTGS2 (0.64) PTGS2FBP1ABL1EGFRABL2
SCHEMBL7104672 0.81 FBP1 (0.60) FBP1ABL1EGFRABL2ALDH1A1
SCHEMBL7104674 0.81 FBP1 (0.60) FBP1ABL1EGFRABL2ALDH1A1
SCHEMBL2748717 0.79 MAOB (0.63) FBP1ALDH1A1KMT2AMEN1
SCHEMBL2748716 0.79 MAOB (0.63) FBP1ALDH1A1KMT2AMEN1
SCHEMBL2748715 0.79 MAOB (0.63) FBP1ALDH1A1KMT2AMEN1
SCHEMBL1959473 0.78 CYSLTR2 (0.57) CYSLTR2CYSLTR1PTGS2ALDH1A1CYP1A2
SCHEMBL8625069 0.76 FBP1 (0.66) PTGS2FBP1ABL1EGFRABL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0023385-B1 ETHANAMINE DERIVATIVES, THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS BEECHAM GROUP PLC (GB) 1982-12-15 EP disclosed
US-4338333-A ANTIOBESITY, HYPOGLYCEMIC BEECHAM GROUP LIMITED (GB) 1982-07-06 US disclosed
EP-0023385-A1 Ethanamine derivatives, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-02-04 EP disclosed