SCHEMBL11264159

SCHEMBL11264159

O=C(NCC1CN=C(c2ccccc2)c2cc(C[N+](=O)[O-])ccc2N1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 8/20 0.56
HPGD P15428 2/20 0.36
LMNA P02545 1/20 0.36
PDE4D Q08499 1/20 0.36
OPRD1 P41143 2/20 0.36
CHRM1 P11229 1/20 0.36
ADRB1 P08588 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
TTK P33981 1/20 0.33
POLB P06746 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10963912 0.83 OPRK1 (0.79) OPRK1HPGDOPRD1ADRB1
SCHEMBL10963938 0.82 OPRK1 (0.41) OPRK1HPGDLMNAPDE4DCHRM1
SCHEMBL11147029 0.69 OPRK1 (0.81) OPRK1HPGDLMNAOPRD1HTT
SCHEMBL10969329 0.68 LMNA (0.58) OPRK1HPGDLMNAPDE4DCHRM1
SCHEMBL10965338 0.66 OPRK1 (0.68) OPRK1LMNAOPRD1
SCHEMBL11352761 0.66 OPRK1 (0.42) OPRK1HPGDLMNAPDE4DCHRM1
SCHEMBL11395623 0.64 OPRK1 (0.40) OPRK1HPGDLMNAPDE4DCHRM1
SCHEMBL10966464 0.63 OPRK1 (0.70) OPRK1OPRD1
SCHEMBL10861062 0.62 CCKBR (0.67) OPRK1OPRD1
SCHEMBL10964736 0.61 OPRK1 (0.66) OPRK1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0054839-A2 2-Acylaminomethyl-1,4-benzodiazepines and their salts, methods of preparing them and pharmaceutical compositions containing them Kali-Chemie Pharma GmbH (DE) 1982-06-30 EP disclosed