SCHEMBL11264210

SCHEMBL11264210

CCCN1CCC[C@H]2CC(O)CC[C@@H]21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.44
DRD1 P21728 2/20 0.44
DRD3 P35462 3/20 0.42
LMNA P02545 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
ADRB2 P07550 1/20 0.42
THRB P10828 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
DRD4 P21917 1/20 0.42
HTR2A P28223 1/20 0.42
CYP2C19 P33261 1/20 0.42
GRM5 P41594 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
BLM P54132 2/20 0.41
CYP3A4 P08684 2/20 0.40
MAPT P10636 2/20 0.40
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11264207 1.00 DRD2 (0.44) DRD2DRD1DRD3LMNAMEN1
SCHEMBL26616920 0.87 DRD2 (0.44) DRD2DRD1DRD3LMNAMEN1
SCHEMBL17538370 0.78 DRD2 (0.51) DRD2DRD1DRD3LMNAMEN1
SCHEMBL11088237 0.78 CYP3A4 (0.39) DRD2DRD1CYP3A4MAPT
SCHEMBL11088225 0.78 CYP3A4 (0.39) DRD2DRD1CYP3A4MAPT
SCHEMBL10839126 0.78 DRD2 (0.40) DRD2DRD1DRD3LMNAMEN1
SCHEMBL11075113 0.77 L3MBTL3 (0.40) DRD2LMNACYP3A4MAPT
SCHEMBL11075108 0.77 L3MBTL3 (0.40) DRD2LMNACYP3A4MAPT
SCHEMBL10839988 0.75 SLC18A3 (0.36) DRD2
SCHEMBL9824261 0.75 SLC18A3 (0.36) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4311844-A Octahydro-2H-pyrrolo[3,4,-g]quinolines ELI LILLY AND COMPANY (US) 1982-01-19 US disclosed
US-4282362-A TREATING PARKINSON'S DISEASE, INHIBITORS OF PRE ACTIN SECRETION, DOPAMINE ANTAGONISTS ELI LILLY AND COMPANY (US) 1981-08-04 US disclosed
US-4235909-A DOPAMINE ANTAGONISTS, IN THE TREATMENT OF PARKINSON'S DISEASE ELI LILLY AND COMPANY (US) 1980-11-25 US disclosed
EP-0013788-A1 Octahydro-2H-pyrrolo(3,4-g)quinolines, process for their preparation and pharmaceutical compositions containing them ELI LILLY AND COMPANY (US) 1980-08-06 EP disclosed