SCHEMBL1126428

SCHEMBL1126428

Cc1cc(C)nc(N2CCN(c3ccc(NC(=O)C(=O)c4ccc(CCC(C)c5ccccc5)[nH]4)cc3)CC2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.37
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
CCR3 P51677 1/20 0.36
MAPT P10636 4/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC2A1 P11166 2/20 0.36
KCNQ2 O43526 1/20 0.35
DRD4 P21917 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
POLB P06746 2/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127189 0.90 CASR (0.35) CASRPSEN1PSEN2APH1BNCSTN
SCHEMBL1126449 0.80 MAPT (0.41) MAPTCYP1A2CYP3A4CYP2D6LMNA
SCHEMBL1127598 0.74 DRD4 (0.39) CASRPSEN1PSEN2APH1BNCSTN
SCHEMBL1987967 0.73 MAPT (0.41) MAPTCYP1A2CYP3A4CYP2D6SLC2A1
SCHEMBL1993235 0.73 KCNQ2 (0.36) CASRPSEN1PSEN2APH1BNCSTN
SCHEMBL1126906 0.73 GAA (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1989517 0.72 MAPT (0.42) MAPTDRD4LMNASMN1; SMN2
SCHEMBL1988341 0.72 DRD4 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1127154 0.72 LMNA (0.36) MAPTCYP1A2CYP3A4CYP2D6LMNA
SCHEMBL1127435 0.72 MAPT (0.40) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed