SCHEMBL11265307

SCHEMBL11265307

COC(=O)C(C(C)=O)C(C(C(=O)OC(C)C)=[N+]([O-])O)c1ccccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
ABCB11 O95342 2/20 0.34
CYP2C19 P33261 2/20 0.34
THRB P10828 1/20 0.34
NR1I2 O75469 1/20 0.34
CHRM2 P08172 1/20 0.34
ADRA2A P08913 1/20 0.34
CYP2B6 P20813 1/20 0.34
DRD1 P21728 1/20 0.34
HTR2A P28223 1/20 0.34
SLC6A4 P31645 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
HTR2B P41595 1/20 0.34
KCNH2 Q12809 1/20 0.34
P2RY12 Q9H244 1/20 0.34
CASP1 P29466 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11393611 1.00 ALDH1A1 (0.36) ALDH1A1ABCB11CYP2C19THRBNR1I2
SCHEMBL11249228 0.91 ALDH1A1 (0.39) ALDH1A1ABCB11CYP2C19THRBNR1I2
Ozone SCHEMBL11388736 0.87 ALDH1A1 (0.36) ALDH1A1ABCB11CYP2C19THRBNR1I2
SCHEMBL11269399 0.83 ALDH1A1 (0.33) ALDH1A1OPRM1
SCHEMBL11387494 0.83 ALDH1A1 (0.33) ALDH1A1OPRM1
SCHEMBL11390896 0.76 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2GAA
SCHEMBL11256342 0.76 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2GAA
SCHEMBL11381249 0.76 ALDH1A1 (0.44) ALDH1A1CYP2C19LMNASMN1; SMN2GAA
SCHEMBL11381243 0.76 ALDH1A1 (0.44) ALDH1A1CYP2C19LMNASMN1; SMN2GAA
SCHEMBL11254194 0.75 ALDH1A1 (0.39) ALDH1A1LMNAGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0009560-A1 1,4-Dihydropyridazine-3-carbonyl compounds, process for their preparation, the compounds for use in curing diseases, medicaments containing them and process for the preparation of the medicaments BAYER AG (DE) 1980-04-16 EP claimed
EP-0009560-B1 1,4-DIHYDROPYRIDAZINE-3-CARBONYL COMPOUNDS, PROCESS FOR THEIR PREPARATION, THE COMPOUNDS FOR USE IN CURING DISEASES, MEDICAMENTS CONTAINING THEM AND PROCESS FOR THE PREPARATION OF THE MEDICAMENTS BAYER AG (DE) 1982-09-22 EP disclosed
US-4280998-A 1,4-Dihydropyridazine-3-carboxylic acid derivatives, a process for their preparation and their use as antihypertensives BAYER AKTIENGESELLSCHAFT (DE) 1981-07-28 US disclosed