SCHEMBL11266822

SCHEMBL11266822

CC(=O)NC(=O)CSC(=O)c1ccc2ncccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.53
HTT P42858 1/20 0.53
PLK1 P53350 1/20 0.53
ALDH1A1 P00352 5/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
TSHR P16473 1/20 0.51
HSD17B10 Q99714 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 1/20 0.46
DOT1L Q8TEK3 1/20 0.45
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
POLB P06746 2/20 0.44
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
GAA P10253 2/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
MAPT P10636 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL359531 0.74 ALOX15 (0.69) ALOX15HTTPLK1ALDH1A1SMN1; SMN2
SCHEMBL29924709 0.74 ALOX15 (0.69) ALOX15HTTPLK1ALDH1A1SMN1; SMN2
SCHEMBL2270839 0.73 ALOX15 (0.64) ALOX15HTTPLK1ALDH1A1SMN1; SMN2
SCHEMBL11264480 0.72 KMT2A (0.60) ALOX15HTTALDH1A1CYP3A4TSHR
SCHEMBL13844834 0.71 PLK1 (0.74) ALOX15HTTPLK1ALDH1A1SMN1; SMN2
SCHEMBL11267948 0.71 MAPT (0.51) HTTALDH1A1SMN1; SMN2LMNANPC1
SCHEMBL27856105 0.70 DOT1L (0.73) ALOX15HTTPLK1ALDH1A1CYP3A4
SCHEMBL2696504 0.70 PTPN1 (0.60) ALOX15HTTPLK1ALDH1A1TSHR
SCHEMBL11962154 0.70 PLK1 (1.00) ALOX15HTTPLK1ALDH1A1SMN1; SMN2
SCHEMBL4402960 0.70 ALOX15 (0.63) ALOX15HTTPLK1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4329363-A Substituted mercapto acid amides and their use MERCK & CO., INC. (US) 1982-05-11 US disclosed
US-4216160-A IMMUNOREGULANTS FOR CORRECTING AN INBALANCE OF IMMUNE HOMEOSTASIS MERCK & CO., INC. (US) 1980-08-05 US disclosed