SCHEMBL11264480

SCHEMBL11264480

CC(=O)NC(=O)CSC(=O)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.60
ALDH1A1 P00352 6/20 0.60
MAPT P10636 5/20 0.60
GPR139 Q6DWJ6 1/20 0.59
L3MBTL1 Q9Y468 2/20 0.49
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.42
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
TSHR P16473 1/20 0.40
POLB P06746 1/20 0.40
KDM4E B2RXH2 2/20 0.39
CES1 P23141 2/20 0.39
MEN1 O00255 1/20 0.39
CYP3A4 P08684 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11267948 0.91 MAPT (0.51) KMT2AALDH1A1MAPTGPR139L3MBTL1
SCHEMBL12642206 0.82 GPR139 (0.62) KMT2AALDH1A1MAPTGPR139L3MBTL1
SCHEMBL9371115 0.81 ALDH1A1 (0.51) KMT2AALDH1A1MAPTGPR139L3MBTL1
SCHEMBL11266779 0.79 KMT2A (0.40) KMT2AALDH1A1MAPTGPR139L3MBTL1
SCHEMBL11267199 0.78 SMN1; SMN2 (0.44) KMT2AALDH1A1MAPTHTTSMN1; SMN2
SCHEMBL9129277 0.77 ALDH1A1 (0.75) KMT2AALDH1A1MAPTGPR139L3MBTL1
SCHEMBL11259579 0.77 PAM (0.62) KMT2AALDH1A1L3MBTL1KDM4ECES1
SCHEMBL8980464 0.77 GPR139 (0.60) KMT2AALDH1A1MAPTGPR139L3MBTL1
SCHEMBL16088012 0.76 KMT2A (0.50) KMT2AALDH1A1MAPTGPR139L3MBTL1
SCHEMBL10101151 0.76 KMT2A (0.56) KMT2AALDH1A1MAPTGPR139L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4329363-A Substituted mercapto acid amides and their use MERCK & CO., INC. (US) 1982-05-11 US disclosed
US-4216160-A IMMUNOREGULANTS FOR CORRECTING AN INBALANCE OF IMMUNE HOMEOSTASIS MERCK & CO., INC. (US) 1980-08-05 US disclosed
EP-0001989-A1 Substituted mercapto acid amides, process for their preparation, pharmaceutical composition containing same and their use MERCK & CO. INC. (US) 1979-05-30 EP disclosed