SCHEMBL1126989

SCHEMBL1126989

COCCn1ccc(-c2cccc(Cl)c2)c1C(=O)C(=O)Cl

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TP53 P04637 1/20 0.39
CHRM3 P20309 7/20 0.38
P2RX7 Q99572 1/20 0.38
HPGD P15428 1/20 0.37
EGFR P00533 2/20 0.36
CECR2 Q9BXF3 1/20 0.36
CNR2 P34972 1/20 0.36
CNR1 P21554 1/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
SLC6A9 P48067 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127046 0.87 CNR1 (0.46) ALDH1A1HPGDCNR2CNR1
SCHEMBL15162449 0.85 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP3A4ALOX15CASP1
SCHEMBL16588815 0.85 TP53 (0.39) ALDH1A1CYP1A2CYP3A4ALOX15CASP1
SCHEMBL1126908 0.80 ALDH1A1 (0.38) ALDH1A1CHRM3P2RX7HPGDCNR2
SCHEMBL1989510 0.78 CNR1 (0.41) ALDH1A1CYP1A2CYP3A4ALOX15CASP1
SCHEMBL1127699 0.76 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP3A4CASP1HSD17B10
SCHEMBL1126995 0.74 GFER (0.39) ALDH1A1CYP1A2CYP3A4HPGDEGFR
SCHEMBL1126629 0.71 ACACB (0.37) ALDH1A1CASP1HSD17B10TP53P2RX7
SCHEMBL15161955 0.71 SMN1; SMN2 (0.44) ALDH1A1CNR2CNR1
SCHEMBL16588838 0.70 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP3A4ALOX15CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed