SCHEMBL1126995

SCHEMBL1126995

COCn1ccc(-c2ccccc2)c1C(=O)C(=O)Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.39
KDM4E B2RXH2 7/20 0.38
ALDH1A1 P00352 5/20 0.38
MAPK1 P28482 1/20 0.38
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
THRB P10828 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CYP2C19 P33261 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
EGFR P00533 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127046 0.86 CNR1 (0.46) GFERKDM4EALDH1A1MAPK1CNR1
SCHEMBL15162305 0.84 KDM4E (0.46) KDM4EALDH1A1MAPK1CNR2SMN1; SMN2
SCHEMBL1127023 0.79 ALDH1A1 (0.58) KDM4EALDH1A1SMN1; SMN2CYP2C19KMT2A
SCHEMBL1126911 0.78 HTR2C (0.41) KDM4EALDH1A1MAPK1CNR2SMN1; SMN2
SCHEMBL15162449 0.75 ALDH1A1 (0.42) KDM4EALDH1A1MAPK1CNR1CNR2
SCHEMBL15162319 0.74 THRB (0.36) GFERKDM4EALDH1A1THRBSMN1; SMN2
SCHEMBL1126989 0.74 ALDH1A1 (0.39) ALDH1A1CNR1CNR2CYP1A2CYP3A4
SCHEMBL1988726 0.72 CCNC (0.40) GFERKDM4EALDH1A1MAPK1CNR1
SCHEMBL1126908 0.71 ALDH1A1 (0.38) KDM4EALDH1A1CNR1CNR2KMT2A
SCHEMBL15161955 0.69 SMN1; SMN2 (0.44) KDM4EALDH1A1CNR1CNR2THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed