SCHEMBL1127007

SCHEMBL1127007

CCc1nc2c(C(F)(F)F)cccc2c(-c2ccccc2)c1C(=O)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 17/20 0.60
NR1H3 Q13133 16/20 0.60
ESR1 P03372 1/20 0.48
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
FABP3 P05413 1/20 0.44
FABP4 P15090 1/20 0.44
FABP5 Q01469 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1125943 0.84 GAA (0.64) NR1H2NR1H3ESR1GAAMAPT
SCHEMBL11043805 0.77 P2RX3 (0.41) NR1H2NR1H3ESR1FABP3FABP4
SCHEMBL6024428 0.75 ESR1 (0.51) NR1H2NR1H3ESR1GAAMAPT
SCHEMBL1124681 0.75 NR1H2 (1.00) NR1H2NR1H3MAPTNPSR1
SCHEMBL1125732 0.73 NR1H2 (0.81) NR1H2NR1H3
SCHEMBL1124620 0.73 NR1H2 (0.81) NR1H2NR1H3
SCHEMBL1124692 0.73 NR1H2 (0.95) NR1H2NR1H3MAPTNPSR1
SCHEMBL1125782 0.72 NR1H2 (0.78) NR1H2NR1H3
SCHEMBL2821238 0.71 FABP4 (0.46) GAAMAPTNPSR1FABP3FABP4
SCHEMBL10946606 0.71 KDM4E (0.46) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2284157-A1 Quinolines useful in treating cardiovascular disease Wyeth (US) 2011-02-16 EP claimed