SCHEMBL6024428

SCHEMBL6024428

Cc1nc2c(C(F)(F)F)cccc2c(-c2ccccc2)c1C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.51
NR1H2 P55055 2/20 0.51
NR1H3 Q13133 2/20 0.51
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
TACR1 P25103 2/20 0.45
ALDH1A1 P00352 4/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP3A4 P08684 1/20 0.42
CD38 P28907 1/20 0.42
ENPP1 P22413 1/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
FABP3 P05413 1/20 0.41
FABP4 P15090 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1125943 0.88 GAA (0.64) ESR1NR1H2NR1H3GAAMAPT
SCHEMBL3855505 0.82 NR1H2 (0.48) ESR1NR1H2NR1H3GAAALDH1A1
SCHEMBL2821537 0.81 GAA (0.45) ESR1NR1H2NR1H3GAAMAPT
SCHEMBL4307232 0.76 NR1H2 (0.43) NR1H2NR1H3GAAMAPTNPSR1
SCHEMBL4012785 0.75 NR1H2 (0.42) ESR1NR1H2NR1H3CYP3A4CD38
SCHEMBL11045513 0.75 ALDH1A1 (0.45) ESR1NR1H2NR1H3ALDH1A1L3MBTL1
SCHEMBL1127007 0.75 NR1H2 (0.60) ESR1NR1H2NR1H3GAAMAPT
SCHEMBL2821849 0.74 GAA (0.46) ESR1NR1H2NR1H3GAAMAPT
SCHEMBL4011398 0.74 NR1H2 (0.49) ESR1NR1H2NR1H3
Hydrochloric Acid SCHEMBL11617104 0.74 ALDH1A1 (0.44) ESR1NR1H2NR1H3ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1692111-A2 QUINOLINES USEFUL IN TREATING CARDIOVASCULAR DISEASE Wyeth, A Corporation of the State of Delaware (US) 2006-08-23 EP disclosed
WO-2005058834-A2 QUINOLINES USEFUL IN TREATING CARDIOVASCULAR DISEASE WYETH (US) 2005-06-30 WO disclosed