SCHEMBL1127083

SCHEMBL1127083

C1=CC=C2CC=CN2C=C1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1703443 0.69
SCHEMBL22077231 0.67
SCHEMBL17090769 0.64
SCHEMBL6986494 0.63
SCHEMBL18469318 0.61
SCHEMBL28015655 0.61 MAPT (0.32)
SCHEMBL24865844 0.59 MGLL (0.36)
SCHEMBL11312340 0.59
SCHEMBL13865281 0.59
SCHEMBL346177 0.59 KDM4E (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed
EP-0763036-B1 [a]-ANNELATED PYRROLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCKLE GMBH (DE) 2002-09-11 EP disclosed
EP-0763037-B1 [a]-ANNELATED PYRROLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCKLE GMBH (DE) 2001-11-14 EP disclosed
EP-0763037-A1 [a]-ANNELATED PYRROLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCKLE GMBH (DE) 1997-03-19 EP disclosed
EP-0763036-A1 [a]-ANNELATED PYRROLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCKLE GMBH (DE) 1997-03-19 EP disclosed
WO-1995032972-A1 [a]-ANNELATED PYRROLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCKLE GMBH (DE) 1995-12-07 WO disclosed
WO-1995032970-A1 (a)-ANNELATED PYRROLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCKLE GMBH (DE) 1995-12-07 WO disclosed