SCHEMBL11272068

SCHEMBL11272068

O=C(NC(Cc1ccccc1)C(=O)Nc1ccc(Cl)nc1C(=O)c1ccccc1)OCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.57
CTSL P07711 1/20 0.51
CTSB P07858 1/20 0.51
CTSS P25774 1/20 0.51
CTSK P43235 1/20 0.51
F2 P00734 2/20 0.49
PRSS1 P07477 2/20 0.49
PRSS2 P07478 2/20 0.49
PRSS3 P35030 2/20 0.49
KDM1A O60341 6/20 0.48
MAOA P21397 4/20 0.48
RCOR1 Q9UKL0 3/20 0.48
KDM1B Q8NB78 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
MAOB P27338 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11269675 0.82 NPSR1 (0.39) TACR1
SCHEMBL11269680 0.79 NPSR1 (0.62) KDM1ARCOR1
SCHEMBL7370634 0.75 HDAC8 (0.73) TACR1CTSLCTSBCTSSCTSK
SCHEMBL4171055 0.75 TACR1 (0.61) TACR1CTSLCTSBCTSSCTSK
SCHEMBL7971421 0.73 TACR1 (1.00) TACR1CTSLCTSBCTSSCTSK
SCHEMBL13768104 0.73 CTSL (0.61) TACR1CTSLCTSBCTSSCTSK
SCHEMBL18444606 0.73 KDM1A (0.68) TACR1CTSLCTSBCTSSCTSK
SCHEMBL8083427 0.73 TACR1 (0.71) TACR1CTSLCTSBCTSSCTSK
SCHEMBL4157711 0.72 TACR1 (0.67) TACR1CTSLCTSBCTSSCTSK
SCHEMBL20441472 0.72 CTSL (0.53) TACR1CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE31071-E 6-Aza-3H-1,4-benzodiazepines DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DE) 1982-11-02 US disclosed
US-4008223-A SPASMOLYTIC, ANTIPHLOGISTIC, TRANQUILIZER DEUTSCHE GOLD- UND SILBER-SCHEIDEANSTALT VORMALS ROESSLER (DT) 1977-02-15 US disclosed