SCHEMBL11272202

SCHEMBL11272202

C/N=C(\NC)NC(=N)Nc1c(C)cccc1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.55
DRD2 P14416 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2B P41595 1/20 0.46
PKM P14618 1/20 0.45
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
NFKB1 P19838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11272212 1.00 POLB (0.55) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11287194 0.81 POLB (0.42) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11280869 0.81 POLB (0.84) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11280882 0.81 POLB (0.84) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11284346 0.80 POLB (0.47) POLBDRD2HTR2AHTR2BPKM
Hydrochloric Acid SCHEMBL11562609 0.79 POLB (0.82) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11251266 0.79 ALDH1A1 (0.44) POLBDRD2HTR2AHTR2BPKM
Hydrochloric Acid SCHEMBL11255459 0.77 ALDH1A1 (0.43) POLBDRD2HTR2AHTR2BPKM
SCHEMBL11138510 0.77 LMNA (0.45) POLBALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL8873938 0.76 ALDH1A1 (0.48) POLBDRD2HTR2AHTR2BPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed