SCHEMBL11275324

SCHEMBL11275324

c1ncc2nc3ccc4cc[nH]c4c3cc2n1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.36
TDO2 P48775 2/20 0.35
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
DYRK1A Q13627 1/20 0.33
AHR P35869 1/20 0.32
PIK3CD O00329 1/20 0.31
PIK3CA P42336 1/20 0.31
RAD52 P43351 1/20 0.31
SMARCA2 P51531 1/20 0.31
PIM3 Q86V86 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL450386 0.82 EGFR (0.40) EGFRTDO2IKBKBCHUKDYRK1A
SCHEMBL16896218 0.81 EGFR (0.39) EGFRTDO2IKBKBCHUKDYRK1A
SCHEMBL20657077 0.73 EGFR (0.47) EGFRTDO2PIK3CDPIK3CA
SCHEMBL19518057 0.72 MAPK1 (0.35) EGFRAHRPIM3
SCHEMBL10744986 0.72 LMNA (0.44) EGFRTDO2RAD52
SCHEMBL88355 0.71 KMT2A (0.47) EGFRAHRRAD52SMARCA2
SCHEMBL16416592 0.71 RAD52 (0.31) RAD52SMARCA2PIM3
SCHEMBL28401294 0.71 EGFR (0.44) EGFRTDO2PIK3CDPIK3CA
SCHEMBL23852799 0.68 AHR (0.38) EGFRTDO2IKBKBCHUKDYRK1A
SCHEMBL7744423 0.65 AHR (0.35) AHRPIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0015786-B1 IMIDAZO AND PYRIMIDO-PYRIDO INDOLES, THEIR PREPARATION AND MEDICINES CONTAINING THEM SYNTHELABO (FR) 1982-04-21 EP claimed
EP-0015786-A1 Imidazo and pyrimido-pyrido indoles, their preparation and medicines containing them SYNTHELABO (FR) 1980-09-17 EP claimed
EP-0015786-B1 IMIDAZO AND PYRIMIDO-PYRIDO INDOLES, THEIR PREPARATION AND MEDICINES CONTAINING THEM SYNTHELABO (FR) 1982-04-21 EP disclosed
EP-0015786-B1 IMIDAZO AND PYRIMIDO-PYRIDO INDOLES, THEIR PREPARATION AND MEDICINES CONTAINING THEM SYNTHELABO (FR) 1982-04-21 EP disclosed
EP-0015786-A1 Imidazo and pyrimido-pyrido indoles, their preparation and medicines containing them SYNTHELABO (FR) 1980-09-17 EP disclosed
EP-0015786-A1 Imidazo and pyrimido-pyrido indoles, their preparation and medicines containing them SYNTHELABO (FR) 1980-09-17 EP disclosed
EP-0015786-A1 Imidazo and pyrimido-pyrido indoles, their preparation and medicines containing them SYNTHELABO (FR) 1980-09-17 EP disclosed