SCHEMBL11275893

SCHEMBL11275893

NN(C(=O)C(F)(F)F)c1nncc(-c2ccccc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
IKBKB O14920 1/20 0.36
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 1/20 0.36
ATR Q13535 3/20 0.36
PRKDC P78527 1/20 0.36
MAP2K3 P46734 1/20 0.35
KDM4E B2RXH2 3/20 0.35
HPGD P15428 2/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
MAPT P10636 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11328971 0.82 MEN1 (0.44) MEN1KMT2AIKBKBALDH1A1NPC1
SCHEMBL11264202 0.73 MEN1 (0.64) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL11275588 0.68 MAPT (0.46) MEN1KMT2AIKBKBALDH1A1NPC1
SCHEMBL9298461 0.67 NPSR1 (0.46) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL27833925 0.66 ALDH1A1 (0.45) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL11262954 0.65 CYP11B2 (0.49) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL21938127 0.65 GABRA1 (0.54) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL2325695 0.64 ADORA2A (0.67) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL21938128 0.64 ALDH1A1 (0.49) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL31009002 0.64 ADORA2A (0.67) MEN1KMT2AALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4310551-A Pharmacologically active substituted 1,2,4-triazines DIAMOND SHAMROCK CORPORATION (US) 1982-01-12 US disclosed
US-4251527-A ANTIINFLAMMATORY AGENTS DIAMOND SHAMROCK CORPORATION (US) 1981-02-17 US disclosed
US-4157392-A HYPOTENSIVE AGENTS, ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIPYRETICS AND NERVOUS SYSTEM EFFECTS DIAMOND SHAMROCK CORPORATION (US) 1979-06-05 US disclosed