SCHEMBL11278705

SCHEMBL11278705

CCc1cccc(C)c1NC(=N)NC(=N)NC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
ALOX12 P18054 1/20 0.50
NLRP3 Q96P20 1/20 0.48
HTT P42858 3/20 0.47
HSD17B10 Q99714 2/20 0.47
POLB P06746 2/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
ALOX15 P16050 1/20 0.45
RAB9A P51151 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CHIT1 Q13231 1/20 0.45
PTGS2 P35354 1/20 0.43
CACNA1C Q13936 1/20 0.41
SCN5A Q14524 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11557047 0.91 SCN5A (0.49) ALDH1A1SMN1; SMN2ALOX12NLRP3HTT
SCHEMBL11274843 0.89 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2ALOX12NLRP3HTT
SCHEMBL10615584 0.88 CACNA1C (0.52) ALDH1A1SMN1; SMN2ALOX12NLRP3HTT
SCHEMBL9177252 0.87 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2ALOX12NLRP3HTT
SCHEMBL11287194 0.85 POLB (0.42) ALDH1A1POLBMEN1KMT2AMAPT
SCHEMBL11274661 0.85 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2ALOX12NLRP3HTT
SCHEMBL11271522 0.84 SCN5A (0.40) ALDH1A1NLRP3KDM4EALOX15RAB9A
SCHEMBL6698675 0.84 NLRP3 (0.50) ALDH1A1SMN1; SMN2ALOX12NLRP3HTT
SCHEMBL11284491 0.81 CACNA1C (0.39) ALDH1A1SMN1; SMN2POLBMEN1KMT2A
SCHEMBL11056404 0.81 CACNA1C (0.54) ALDH1A1SMN1; SMN2ALOX12NLRP3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326075-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4203920-A ANTIDIARRHEAL WILLIAM H. RORER, INC. (US) 1980-05-20 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed
US-4060635-A Amidinoureas for treating diarrhea WILLIAM H. RORER, INC. (US) 1977-11-29 US disclosed