SCHEMBL11279308

SCHEMBL11279308

COc1ccc(C(=O)Oc2cc(C(CNC(C)(C)C)OS(C)(=O)=O)ccc2OC(C)=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.44
TP53 P04637 1/20 0.43
GAA P10253 1/20 0.43
THRB P10828 1/20 0.43
CCR5 P51681 2/20 0.43
SLC2A1 P11166 1/20 0.43
ALDH1A1 P00352 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
PKM P14618 1/20 0.39
MAPT P10636 4/20 0.37
MEN1 O00255 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11286085 1.00 KMT2A (0.44) KMT2ATP53GAATHRBCCR5
Alcohol SCHEMBL11290095 0.97 KMT2A (0.42) KMT2ATP53GAATHRBCCR5
Alcohol SCHEMBL11558382 0.88 CCR5 (0.39) KMT2ATP53GAATHRBCCR5
SCHEMBL11286259 0.87 SLC2A1 (0.40) KMT2ATP53GAATHRBSLC2A1
Nisbuterol SCHEMBL11286092 0.87 ADRB3 (0.46) KMT2ATP53GAATHRBCCR5
SCHEMBL11279314 0.87 ADRB3 (0.46) KMT2ATP53GAATHRBCCR5
Alcohol SCHEMBL11286257 0.85 SLC2A1 (0.38) KMT2ATP53GAATHRBSLC2A1
Nisbuterol SCHEMBL29385412 0.84 KMT2A (0.49) KMT2ATP53GAATHRBCCR5
SCHEMBL11284114 0.83 ACHE (0.38) KMT2ATP53GAATHRBALDH1A1
Alcohol SCHEMBL11559195 0.83 KMT2A (0.39) KMT2ATP53GAATHRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4336400-A BRONCHODILATOR AGENTS, CARDIOVASCULAR STIMULANTS STERLING DRUG INC. (US) 1982-06-22 US claimed
US-4336400-A BRONCHODILATOR AGENTS, CARDIOVASCULAR STIMULANTS STERLING DRUG INC. (US) 1982-06-22 US disclosed
US-RE30241-E BRONCHODILATION, ADRENERGIC STIMULANTS STERLING DRUG INC. (US) 1980-03-25 US disclosed
US-4138581-A BRONCHODILATOR AGENTS, ADRENERGIC STIMULANTS STERLING DRUGS INC. (US) 1979-02-06 US disclosed