SCHEMBL11279566

SCHEMBL11279566

CC(CS)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 10/20 0.58
ACE2 Q9BYF1 5/20 0.57
CMA1 P23946 2/20 0.56
HSD17B10 Q99714 2/20 0.55
KDM4E B2RXH2 1/20 0.55
F2 P00734 1/20 0.55
REN P00797 1/20 0.55
LMNA P02545 1/20 0.55
LTA4H P09960 1/20 0.55
MAPT P10636 1/20 0.55
PEPD P12955 1/20 0.55
ALOX15 P16050 1/20 0.55
PTGS1 P23219 1/20 0.55
HTR2A P28223 1/20 0.55
PTGS2 P35354 1/20 0.55
HRH1 P35367 1/20 0.55
THPO P40225 1/20 0.55
PMP22 Q01453 1/20 0.55
CTRB1 P17538 1/20 0.55
SLC6A2 P23975 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7388885 1.00 ACE (0.58) ACEACE2CMA1HSD17B10KDM4E
SCHEMBL7388881 1.00 ACE (0.58) ACEACE2CMA1HSD17B10KDM4E
SCHEMBL11338055 0.94 ACE (0.54) ACEACE2CMA1HSD17B10KDM4E
Alacepril SCHEMBL11458085 0.92 ACE (0.51) ACEACE2CMA1CTRB1SLC6A2
SCHEMBL11334873 0.89 ACE (0.59) ACEACE2CMA1HSD17B10SLC6A2
SCHEMBL11279851 0.88 CMA1 (0.57) ACEACE2CMA1CTRB1
SCHEMBL29868291 0.88 OPRM1 (0.59) F2CTRB1SLC6A2OPRM1
SCHEMBL31184433 0.87 SLC6A2 (0.63) ACECMA1SLC6A2OPRM1
SCHEMBL11091524 0.87 SLC6A2 (0.63) ACECMA1SLC6A2OPRM1
Alacepril SCHEMBL34559 0.86 ACE (0.55) ACEACE2CMA1HSD17B10SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007477-B1 1-(3-MERCAPTO-2-METHYLPROPANOYL)PROLYL AMINO ACID DERIVATIVES AND SALTS THEREOF, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDS Dainippon Pharmaceutical Co., Ltd. (JP) 1982-04-28 EP disclosed
US-4248883-A ANTIHYPERTENSION AGENTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1981-02-03 US disclosed
EP-0007477-A1 1-(3-Mercapto-2-methylpropanoyl)prolyl amino acid derivatives and salts thereof, processes for their preparation, and pharmaceutical compositions containing such compounds Dainippon Pharmaceutical Co., Ltd. (JP) 1980-02-06 EP disclosed