SCHEMBL11279898

SCHEMBL11279898

O=C1N=C(N2CCNCC2)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.54
CHRM2 P08172 3/20 0.47
CHRM4 P08173 3/20 0.47
CHRM5 P08912 3/20 0.47
CHRM1 P11229 3/20 0.47
CHRM3 P20309 3/20 0.47
DRD1 P21728 3/20 0.47
KCNH2 Q12809 3/20 0.47
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
MTOR P42345 2/20 0.47
HTR7 P34969 5/20 0.45
HTR2A P28223 4/20 0.45
HTR6 P50406 3/20 0.45
HTR1A P08908 3/20 0.45
HTR5A P47898 2/20 0.45
HTR3A P46098 2/20 0.44
ADRB1 P08588 2/20 0.44
HTR3E A5X5Y0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14352419 0.79 MEN1 (0.53) CYP1A2KDM4EMEN1ALDH1A1LMNA
SCHEMBL725002 0.78 DRD2 (0.49) DRD2CHRM2CHRM4CHRM5CHRM1
SCHEMBL11119265 0.74 HRH4 (0.45) DRD2HTR7HTR2AHTR6HTR1A
SCHEMBL4431761 0.72 DRD2 (0.57) DRD2CHRM2CHRM4CHRM5CHRM1
SCHEMBL167601 0.71 DRD2 (0.74) DRD2CHRM2CHRM4CHRM5CHRM1
SCHEMBL141985 0.71 HRH4 (0.71) DRD2CHRM2CHRM4CHRM5CHRM1
SCHEMBL3410493 0.71 CHRM1 (0.74) DRD2CHRM2CHRM4CHRM5CHRM1
SCHEMBL29969899 0.71 DRD2 (0.74) DRD2CHRM2CHRM4CHRM5CHRM1
SCHEMBL8311 0.70 DRD2 (1.00) DRD2CHRM2CHRM4CHRM5CHRM1
SCHEMBL29368614 0.70 DRD2 (1.00) DRD2CHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4355031-A 2,3-Dihydro-3-[4-(substituted)-1-piperazinyl]-1H-isoindol-1-ones AMERICAN HOME PRODUCTS CORP. (US) 1982-10-19 US disclosed