SCHEMBL11279926

SCHEMBL11279926

O=C(O)C[C@H](NC(=O)CCS)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.55
CA4 P22748 1/20 0.55
MME P08473 3/20 0.47
EPHX2 P34913 2/20 0.43
GNPAT O15228 1/20 0.42
FOLH1 Q04609 2/20 0.42
RECQL P46063 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
PTGS1 P23219 1/20 0.40
GSTK1 Q9Y2Q3 1/20 0.40
CASP3 P42574 1/20 0.40
MAPT P10636 2/20 0.39
RIMKLA Q8IXN7 1/20 0.39
NAALAD2 Q9Y3Q0 1/20 0.39
KDM4E B2RXH2 1/20 0.39
THRB P10828 1/20 0.39
ALOX15 P16050 1/20 0.39
NFKB1 P19838 1/20 0.39
PTGS2 P35354 1/20 0.39
THPO P40225 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13674348 0.87 CA2 (0.62) CA2CA4MMEEPHX2GNPAT
SCHEMBL11269717 0.85 MEN1 (0.47) CA2CA4GNPATRECQLSMN1; SMN2
SCHEMBL12509112 0.84 GNPAT (0.43) CA2CA4MMEGNPATFOLH1
SCHEMBL15912290 0.84 GNPAT (0.43) CA2CA4MMEGNPATFOLH1
SCHEMBL929193 0.83 KDM4E (0.57) CA2CA4GNPATFOLH1RECQL
SCHEMBL5841326 0.83 CA2 (0.58) CA2CA4MMEEPHX2FOLH1
SCHEMBL4572556 0.83 CA2 (0.58) CA2CA4MMEEPHX2GNPAT
SCHEMBL13654776 0.83 CA2 (0.58) CA2CA4MMEEPHX2GNPAT
SCHEMBL4156554 0.82 FOLH1 (0.62) EPHX2GNPATFOLH1RIMKLANAALAD2
SCHEMBL4156556 0.82 FOLH1 (0.62) EPHX2GNPATFOLH1RIMKLANAALAD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4339600-A ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1982-07-13 US disclosed
US-4199512-A Compounds for alleviating hypertension E. R. SQUIBB & SONS, INC. (US) 1980-04-22 US disclosed
US-4173704-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1979-11-06 US disclosed
US-4140786-A ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1979-02-20 US disclosed
US-4140797-A MERCAPTOACYL AMINO ACIDS, ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1979-02-20 US disclosed
US-4112119-A MERCAPTOACYL AMINOACIDS E. R. SQUIBB & SONS, INC. (US) 1978-09-05 US disclosed
US-4053651-A MERCAPTOACYL AMINO ACIDS, ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1977-10-11 US disclosed