Bromide

Bromide

SCHEMBL11279935

Br.COC(=O)c1ccccc1NC(=O)c1sc(N)nc1C

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.98
MAPK1 P28482 3/20 0.98
GAA P10253 2/20 0.98
NPC1 O15118 3/20 0.60
RAB9A P51151 3/20 0.60
KMT2A Q03164 6/20 0.57
HSD17B10 Q99714 4/20 0.57
MEN1 O00255 3/20 0.57
MAPT P10636 3/20 0.57
HPGD P15428 2/20 0.57
ALOX15 P16050 2/20 0.57
HCRTR1 O43613 1/20 0.57
MCL1 Q07820 1/20 0.57
APOBEC3G Q9HC16 1/20 0.57
USP2 O75604 1/20 0.54
CASP1 P29466 1/20 0.54
TSHR P16473 5/20 0.50
LCK P06239 1/20 0.50
KDM4E B2RXH2 1/20 0.50
RXFP1 Q9HBX9 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1540091 0.82 ALDH1A1 (0.70) ALDH1A1MAPK1GAANPC1RAB9A
SCHEMBL3579979 0.80 KMT2A (0.76) ALDH1A1MAPK1GAANPC1RAB9A
SCHEMBL11700991 0.79 KMT2A (0.73) ALDH1A1MAPK1GAANPC1RAB9A
SCHEMBL12335742 0.77 CYP1A2 (0.65) ALDH1A1MAPK1GAAKMT2AHSD17B10
SCHEMBL42334 0.76 RAB9A (0.97) ALDH1A1MAPK1GAANPC1RAB9A
SCHEMBL276275 0.73 ALDH1A1 (0.62) ALDH1A1MAPK1GAANPC1RAB9A
SCHEMBL7721970 0.73 HSD17B10 (0.69) ALDH1A1MAPK1GAANPC1RAB9A
SCHEMBL13186300 0.73 ALDH1A1 (0.58) ALDH1A1MAPK1GAARAB9AKMT2A
SCHEMBL3586328 0.73 RAB9A (0.77) ALDH1A1MAPK1GAANPC1RAB9A
SCHEMBL1540033 0.72 LCK (0.74) ALDH1A1MAPK1GAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-57183768-A None JP disclosed
JP-S57183768-A 4-METHYL-5-(O-CARBOXYPHENYL)CARBAMOYLTHIAZOLE DERIVATIVE AND ITS PREPARATION KANTO ISHI PHARMA CO LTD 1982-11-12 JP disclosed