SCHEMBL276275

SCHEMBL276275

COC(=O)c1sc(N)nc1C

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.62
GAA P10253 1/20 0.57
MAPK1 P28482 1/20 0.57
MAPT P10636 2/20 0.56
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
KMT2A Q03164 1/20 0.51
HPGD P15428 1/20 0.50
LCK P06239 1/20 0.50
CYP1A2 P05177 1/20 0.49
POLB P06746 1/20 0.46
KDM4E B2RXH2 2/20 0.45
PKM P14618 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL244752 0.81 ALDH1A1 (0.73) ALDH1A1MAPTNPC1RAB9AHPGD
SCHEMBL3434838 0.80 ALDH1A1 (0.53) ALDH1A1GAAMAPK1MAPTNPC1
SCHEMBL6985283 0.80 ALDH1A1 (0.53) ALDH1A1GAAMAPK1MAPTNPC1
Hydrochloric Acid SCHEMBL8114168 0.80 ALDH1A1 (0.71) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL10049913 0.80 NPC1 (0.54) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL10532167 0.80 ALDH1A1 (0.49) ALDH1A1GAAMAPK1MAPTNPC1
SCHEMBL10532170 0.80 ALDH1A1 (0.57) ALDH1A1GAAMAPK1MAPTNPC1
SCHEMBL8574686 0.79 KDM4E (0.48) ALDH1A1GAAMAPK1MAPTKMT2A
SCHEMBL8146643 0.79 KDM4E (0.48) ALDH1A1GAAMAPK1MAPTKMT2A
SCHEMBL20911243 0.78 ALDH1A1 (0.76) ALDH1A1GAAMAPK1MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 113 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4288362-A Monoazo pigments containing a quinazo linonylacetoacetanilide coupling component BAYER AKTIENGESELLSCHAFT (DE) 1981-09-08 US claimed
US-12545654-B2 MYC inhibitors and uses thereof STEMSYNERGY THERAPEUTICS, INC. (US) 2026-02-10 US disclosed
EP-4578451-A2 COMPOUNDS AND COMPOSITIONS AS SPPL2A INHIBITORS Novartis AG (CH) 2025-07-02 EP disclosed
EP-4214210-B1 COMPOUNDS AND COMPOSITIONS AS SPPL2A INHIBITORS NOVARTIS AG (CH) 2025-04-09 EP disclosed
US-20250084074-A1 SUBSTITUTED HETEROCYCLES AS HSET INHIBITORS MERCK PATENT GMBH (DE) 2025-03-13 US disclosed
CN-119421877-A Substituted heterocyclic compounds as HSET inhibitors 默克专利股份公司 2025-02-11 CN disclosed
EP-4463444-A1 SUBSTITUTED HETEROCYCLES AS HSET INHIBITORS Merck Patent GmbH (DE) 2024-11-20 EP disclosed
US-20230365571-A1 COMPOUNDS AND COMPOSITIONS AS Sppl2a INHIBITORS NOVARTIS AG (CH) 2023-11-16 US disclosed
US-20230365571-A1 COMPOUNDS AND COMPOSITIONS AS Sppl2a INHIBITORS NOVARTIS AG (CH) 2023-11-16 US disclosed
US-20230365571-A1 COMPOUNDS AND COMPOSITIONS AS Sppl2a INHIBITORS NOVARTIS AG (CH) 2023-11-16 US disclosed
US-4988698-A Cardiovascular disorders, hypotensive agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-01-29 US disclosed
CN-1042905-A The preparation method of 2 (1H) quinolinone compounds and medicinal compositions thereof FUJISAWA PHARMACEUTICAL CO (JP) 1990-06-13 CN disclosed
EP-0370381-A2 2(1H)-quinolinone compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-05-30 EP disclosed
US-4421601-A LACQUERS, INKS, PAINTS, TEXTILES, PAPER BAYER AKTIENGESELLSCHAFT (DE) 1983-12-20 US disclosed
US-4288362-A Monoazo pigments containing a quinazo linonylacetoacetanilide coupling component BAYER AKTIENGESELLSCHAFT (DE) 1981-09-08 US disclosed
US-4260540-A SPIN DYEING POLYACRYLONITRILE BAYER AKTIENGESELLSCHAFT (DE) 1981-04-07 US disclosed
US-4246401-A Axomethine pigments BAYER AKTIENGESELLSCHAFT (DE) 1981-01-20 US disclosed
US-4225489-A Heterocyclic azo dyes and pigments containing 4-quinazolinone moieties BAYER AKTIENGESELLSCHAFT (DE) 1980-09-30 US disclosed
US-4118185-A FASTNESS, DEEP COLORS, AZO DYES, THIAZOLE DYES, PYRIDINE DYES HOECHST AKTIENGESELLSCHAFT (DE) 1978-10-03 US disclosed
US-4014863-A LACQUERS, PRINTING INKS, PAINTS BAYER AKTIENGESELLSCHAFT (DT) 1977-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230365571-A1 COMPOUNDS AND COMPOSITIONS AS Sppl2a INHIBITORS SPPL2A, SPPL2B, BACE1 ALDH1A1 3565/4885GAA 2507/4885MAPK1 1689/4885
US-20250084074-A1 SUBSTITUTED HETEROCYCLES AS HSET INHIBITORS VHL, CDKN1A, CCNI ALDH1A1 1680/4885GAA 1328/4885MAPK1 577/4885
US-12545654-B2 MYC inhibitors and uses thereof MYC, MYCBP, NR2E1 ALDH1A1 4317/4885GAA 4531/4885MAPK1 279/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.