SCHEMBL11280672

SCHEMBL11280672

CC(=O)SCC(C)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 10/20 0.52
PREP P48147 4/20 0.51
ACE P12821 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600176 0.83 FKBP1A (0.41) FKBP1AACE
Hydrochloric Acid SCHEMBL7263625 0.83 FKBP1A (0.56) FKBP1APREPALDH1A1CYP3A4TSHR
SCHEMBL6788131 0.81 FKBP1A (0.64) FKBP1APREPACE
SCHEMBL6788139 0.81 FKBP1A (0.64) FKBP1APREPACE
SCHEMBL11940447 0.81 FKBP1A (0.64) FKBP1APREPACE
SCHEMBL11274848 0.81 CTRB1 (0.52) ACE
SCHEMBL10794593 0.80 ACE (0.59) ACE
SCHEMBL10794601 0.80 ACE (0.59) ACE
SCHEMBL11281963 0.79 CTRB1 (0.47) PREPACETSHR
SCHEMBL11281958 0.79 CTRB1 (0.47) PREPACETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007477-B1 1-(3-MERCAPTO-2-METHYLPROPANOYL)PROLYL AMINO ACID DERIVATIVES AND SALTS THEREOF, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDS Dainippon Pharmaceutical Co., Ltd. (JP) 1982-04-28 EP disclosed
US-4248883-A ANTIHYPERTENSION AGENTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1981-02-03 US disclosed
EP-0007477-A1 1-(3-Mercapto-2-methylpropanoyl)prolyl amino acid derivatives and salts thereof, processes for their preparation, and pharmaceutical compositions containing such compounds Dainippon Pharmaceutical Co., Ltd. (JP) 1980-02-06 EP disclosed