SCHEMBL1128243

SCHEMBL1128243

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nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.38
CTSK P43235 2/20 0.38
AAK1 Q2M2I8 2/20 0.32
MMP13 P45452 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MME P08473 1/20 0.30
ACE P12821 1/20 0.30
CPA1 P15085 1/20 0.30
ACE2 Q9BYF1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL67050 1.00 CTSS (0.38) CTSSCTSKAAK1MMP13KMT2A
SCHEMBL31703376 1.00 CTSS (0.38) CTSSCTSKAAK1MMP13KMT2A
SCHEMBL67051 1.00 CTSS (0.38) CTSSCTSKAAK1MMP13KMT2A
SCHEMBL27645074 1.00 CTSS (0.38) CTSSCTSKAAK1MMP13KMT2A
SCHEMBL1486202 1.00 CTSS (0.38) CTSSCTSKAAK1MMP13KMT2A
SCHEMBL8460615 0.87 CA2 (0.34) CTSSCTSKAAK1MMP13KMT2A
SCHEMBL10273899 0.87 AAK1 (0.32) AAK1MMP13KMT2AMEN1GAA
SCHEMBL28760575 0.85 CTSS (0.38) CTSSCTSKKMT2AMEN1GAA
SCHEMBL11661957 0.85 CTSS (0.38) CTSSCTSKKMT2AMEN1GAA
SCHEMBL11661955 0.85 CTSS (0.38) CTSSCTSKKMT2AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283009-A1 INHIBITORS OF JNK F. Hoffmann-La Roche AG (CH) 2011-02-16 EP claimed
WO-2009138340-A1 INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2009-11-19 WO claimed
CN-102037092-A Amino acid generator and polysiloxane composition containing the same NISSAN CHEMICAL IND LTD 2011-04-27 CN disclosed
EP-2283009-A1 INHIBITORS OF JNK F. Hoffmann-La Roche AG (CH) 2011-02-16 EP disclosed
WO-2009138340-A1 INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2009-11-19 WO disclosed