SCHEMBL11283641

SCHEMBL11283641

O=C(c1cccnc1)C(F)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
APP P05067 1/20 0.55
GAA P10253 1/20 0.55
HCAR3 P49019 1/20 0.55
HCAR2 Q8TDS4 1/20 0.55
PLOD2 O00469 1/20 0.51
EPHX2 P34913 2/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HTT P42858 1/20 0.49
F7 P08709 1/20 0.49
F3 P13726 1/20 0.49
SARM1 Q6SZW1 1/20 0.49
SIRT2 Q8IXJ6 1/20 0.49
SIRT6 Q8N6T7 1/20 0.49
SIRT1 Q96EB6 1/20 0.49
SIRT3 Q9NTG7 1/20 0.49
SIRT5 Q9NXA8 1/20 0.49
SIRT4 Q9Y6E7 1/20 0.49
LMNA P02545 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4483081 0.82 TDP1 (0.61) ALDH1A1LMNASMN1; SMN2CYP3A4CYP2D6
SCHEMBL11065543 0.81 LMNA (0.67) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL8101551 0.81 MEN1 (0.52) ALDH1A1PLOD2EPHX2CYP2C9CYP2C19
SCHEMBL9292468 0.80 ALDH1A1 (0.59) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL11820789 0.80 ALDH1A1 (0.55) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL7147666 0.80 ALDH1A1 (0.55) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL9603054 0.80 ALDH1A1 (0.55) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL6203223 0.80 ALDH1A1 (0.55) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL27566013 0.79 ALDH1A1 (0.58) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL30641184 0.79 ALDH1A1 (0.57) ALDH1A1APPGAAHCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0008755-B1 ANTIINFLAMMATORY 4,5-DIARYL-2-NITROIMIDAZOLES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-04-21 EP disclosed
US-4251535-A ANTIARTHRITIC AGENTS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1981-02-17 US disclosed
US-4199592-A Antiinflammatory 4,5-diaryl-2-nitroimidazoles E. I. DU PONT DE NEMOURS AND COMPANY (US) 1980-04-22 US disclosed
EP-0008755-A1 Antiinflammatory 4,5-diaryl-2-nitroimidazoles, method for their preparation and pharmaceutical composition containing them E.I. DU PONT DE NEMOURS AND COMPANY (US) 1980-03-19 EP disclosed