SCHEMBL7147666

SCHEMBL7147666

O=C(c1cccnc1)C(Br)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
APP P05067 1/20 0.55
GAA P10253 1/20 0.55
HCAR3 P49019 1/20 0.55
HCAR2 Q8TDS4 1/20 0.55
PLOD2 O00469 1/20 0.51
EPHX2 P34913 2/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HTT P42858 1/20 0.49
F7 P08709 1/20 0.49
F3 P13726 1/20 0.49
SARM1 Q6SZW1 1/20 0.49
SIRT2 Q8IXJ6 1/20 0.49
SIRT6 Q8N6T7 1/20 0.49
SIRT1 Q96EB6 1/20 0.49
SIRT3 Q9NTG7 1/20 0.49
SIRT5 Q9NXA8 1/20 0.49
SIRT4 Q9Y6E7 1/20 0.49
CES2 O00748 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6546257 0.98 ALDH1A1 (0.53) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL7140967 0.90 SMN1; SMN2 (0.51) ALDH1A1APPGAAHCAR3HCAR2
Bromide SCHEMBL6282444 0.89 SMN1; SMN2 (0.50) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL627867 0.82 CES2 (0.64) ALDH1A1HTTCES2CES1LMNA
SCHEMBL11065543 0.81 LMNA (0.67) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL3115655 0.81 MEN1 (0.52) ALDH1A1PLOD2EPHX2CYP2C9CYP2C19
SCHEMBL19104771 0.81 CES2 (0.53) ALDH1A1PLOD2EPHX2CYP2C9CYP2C19
SCHEMBL7262916 0.80 ALDH1A1 (0.59) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL11283641 0.80 ALDH1A1 (0.55) ALDH1A1APPGAAHCAR3HCAR2
SCHEMBL11820789 0.80 ALDH1A1 (0.55) ALDH1A1APPGAAHCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620825-B1 1,3-Azole compound substituted by pyridyl; administering as antiasthmatic, antiinflammatory or antiallergen agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-16 US disclosed
US-6436966-B1 Adenosine A3 receptor antagonists TAKEDA CHEMICAL IND., LTD. (JP) 2002-08-20 US disclosed
WO-1983002613-A1 TRISUBSTITUTED OXAZO COMPOUNDS SALLMANN, ALFRED 1983-08-04 WO disclosed
EP-0084756-A1 Trisubstituted oxaza compounds CIBA-GEIGY AG (CH) 1983-08-03 EP disclosed
EP-0082111-A2 Process for the preparation of imidazoles CIBA-GEIGY AG (CH) 1983-06-22 EP disclosed
EP-0046451-A2 Diaryl-imidazole compounds, methods for their preparation, pharmaceutical drugs containing them and their use CIBA-GEIGY AG (CH) 1982-02-24 EP disclosed