SCHEMBL11287202

SCHEMBL11287202

CSc1ccc(Nc2ncc([N+](=O)[O-])c(O)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
MAPT P10636 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 1/20 0.53
MCL1 Q07820 1/20 0.53
PTK2B Q14289 1/20 0.53
GSK3B P49841 7/20 0.51
GSK3A P49840 5/20 0.51
AURKA O14965 5/20 0.51
SYK P43405 1/20 0.45
STK17A Q9UEE5 1/20 0.42
PLK1 P53350 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TRPV1 Q8NER1 1/20 0.40
STK3 Q13188 1/20 0.40
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11193854 0.85 PTK2B (0.48) MEN1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL5407955 0.84 GSK3B (0.59) MEN1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL11348508 0.82 GSK3B (0.72) MEN1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL11291261 0.82 MAPT (0.53) MEN1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL11287006 0.81 MEN1 (0.52) MEN1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL3580667 0.77 SYK (0.46) MEN1MAPTKMT2AGSK3BAURKA
SCHEMBL11187199 0.77 MEN1 (0.47) MEN1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL11179027 0.75 GSK3B (0.47) MEN1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL17446345 0.74 PIN1 (0.70) MEN1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL10680837 0.71 KMT2A (0.45) MEN1CYP1A2CYP3A4MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0051773-A1 Penicillins, their salts, process for their preparation and pharmaceutical compositions containing them Dr. Karl Thomae GmbH (DE) 1982-05-19 EP disclosed