SCHEMBL11287291

SCHEMBL11287291

Cc1c(C(=O)O)sc2ccc(Cc3ncc[nH]3)cc12

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 4/20 0.55
GPR35 Q9HC97 1/20 0.44
TAAR1 Q96RJ0 3/20 0.43
ROCK1 Q13464 6/20 0.42
HTR1A P08908 1/20 0.36
RXFP1 Q9HBX9 2/20 0.36
PKM P14618 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PRNP P04156 1/20 0.34
BCAT2 O15382 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10955250 0.91 TBXAS1 (0.55) TBXAS1GPR35TAAR1ROCK1HTR1A
SCHEMBL10953653 0.87 ROCK1 (0.45) TBXAS1TAAR1ROCK1
SCHEMBL10952018 0.81 TBXAS1 (0.53) TBXAS1GPR35TAAR1RXFP1PKM
SCHEMBL10953013 0.78 TBXAS1 (0.42) TBXAS1TAAR1ROCK1HTR1ANPSR1
SCHEMBL149468 0.78 TBXAS1 (0.54) TBXAS1TAAR1ROCK1HTR1A
Hydrochloric Acid SCHEMBL10853856 0.77 TBXAS1 (0.53) TBXAS1TAAR1ROCK1HTR1A
SCHEMBL9613211 0.76 TBXAS1 (0.60) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL10948748 0.76 TBXAS1 (0.60) TBXAS1GPR35ROCK1RXFP1PKM
SCHEMBL9757026 0.75 TBXAS1 (0.58) TBXAS1GPR35ROCK1RXFP1PKM
SCHEMBL11168704 0.71 TBXAS1 (0.41) TBXAS1TAAR1ROCK1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0050957-A1 Heterocyclic thromboxane synthetase inhibitors, processes for their preparation, and pharmaceutical compositions containing them Pfizer Limited (GB) 1982-05-05 EP disclosed